Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GODHBSJSHXUGIE
|
8.1 | IC50 | 3 | — | |
SHKVYTQIJOOEMA
|
8.1 | IC50 | 6 | — | |
NHHQJBCNYHBUSI
|
8.0 | Kd | 220 | — | |
VEVUBFZLKUNGER
|
8.0 | IC50 | 3 | — | |
KCVMRCBFSCVBTH
|
8.0 | IC50 | 3 | Yes | |
WNMAXXDDBQOLPI
|
8.0 | IC50 | 5 | — | |
IWBIEKJAAQYGMI
|
8.0 | IC50 | 3 | — | |
BQUCMYBIGNGMFC
|
8.0 | IC50 | 5 | — | |
BYYOHNRGQACTPJ
|
8.0 | IC50 | 2 | — | |
CUDVHEFYRIWYQD
|
8.0 | IC50 | 11 | — | |
DUZZUNRKDFGPSJ
|
8.0 | IC50 | 5 | — | |
IZRLUPFLGZEWCW
|
8.0 | IC50 | 2 | — | |
KUZBKIYSYFCFOT
|
8.0 | IC50 | 5 | — | |
QCTUWJMAPLGTOR
|
8.0 | IC50 | 5 | — | |
XCHWBXBDZRJVDP
|
8.0 | Ki | 51 | — | |
FUNGTOAZDDISQB
|
8.0 | IC50 | 4 | Yes | |
JXDYOSVKVSQGJM
|
8.0 | IC50 | 7 | — | |
XZJHYNMIHBWFCD
|
8.0 | IC50 | 3 | — | |
HUBJRBJFRJHZIG
|
7.9 | IC50 | 3 | — | |
MMCWBZCSGNCOMQ
|
7.9 | IC50 | 5 | Yes | |
CFIBXVQLBVNOHW
|
7.9 | Ki | 64 | — | |
HRZOUBQYVUXBNS
|
7.9 | Ki | 38 | — | |
KNACLJBHKVSTDL
|
7.9 | Ki | 40 | — | |
UXQLMVSZSYZFID
|
7.9 | Ki | 12 | — | |
DZSUJUOJJJCWGG
|
7.9 | IC50 | 55 | Yes | |
JZCBGMAKTMOCFP
|
7.9 | IC50 | 4 | Yes | |
NNAMXKXTCQOZGS
|
7.9 | IC50 | 5 | Yes | |
VOEBMPAZQQYYGC
|
7.9 | IC50 | 5 | Yes | |
XZXHXSATPCNXJR
|
7.9 | IC50 | 165 | Yes | |
HQRUNGNEQLUCLO
|
7.9 | IC50 | 2 | — | |
VDXARSHJPFZWJT
|
7.9 | IC50 | 2 | — | |
FAYAUAZLLLJJGH
|
7.8 | IC50 | 36 | Yes | |
FYLZILJOKOVUAW
|
7.8 | IC50 | 3 | — | |
QCOBLDQZJWXXDC
|
7.8 | IC50 | 2 | — | |
KRIUNPBAQZGFQA
|
7.8 | Ki | 76 | — | |
MPVGZUGXCQEXTM
|
7.8 | IC50 | 61 | Yes | |
PCIMPOMGHFNGMS
|
7.8 | IC50 | 7 | — | |
YCIIZJUIBNPNED
|
7.8 | IC50 | 2 | — | |
YDWMUCKJUNLURC
|
7.8 | Ki | 24 | — | |
YHVHYWYQEFELOW
|
7.8 | IC50 | 44 | — | |
CPTVWYCNJGYSDW
|
7.8 | IC50 | 3 | — | |
BPXQYAXTDCQZHB
|
7.8 | IC50 | 7 | Yes | |
NMJILYFXNANMKC
|
7.8 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
IHJBFEQZLKXMGF
|
7.8 | IC50 | 3 | — | |
BLAFVGLBBOPRLP
|
7.8 | IC50 | 7 | Yes | |
VLXIXYDIKYYMAQ
|
7.8 | IC50 | 7 | — | |
VOYMOBPSYVKQGF
|
7.8 | IC50 | 3 | — | |
HMZRSZQIXPNKJY
|
7.7 | IC50 | 4 | — | |
AAVVJYRIFZWOQJ
|
7.7 | IC50 | 3 | — |