Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PIBOSMWVYTUUIX
|
8.3 | IC50 | 3 | — | |
BIKYDWLMTPRSQL
|
8.3 | Ki | 50 | — | |
CZGMEOAMQWAJOY
|
8.3 | IC50 | 15 | Yes | |
HKZKELVPGXJIMW
|
8.3 | Ki | 41 | — | |
MQRDVGBWWVWMEN
|
8.3 | Ki | 47 | — | |
ONSZEUCTVQJHOZ
|
8.3 | IC50 | 9 | — | |
PWDPLHOKCYLVIC
|
8.3 | IC50 | 5 | — | |
SFPWNTQWFFNJIH
|
8.3 | Ki | 48 | — | |
SILANKVZJSUJHJ
|
8.3 | IC50 | 9 | — | |
UCHQCSDTPQKAKL
|
8.3 | IC50 | 9 | Yes | |
UTZFAVQAWTWOKK
|
8.3 | IC50 | 5 | — | |
YEHCNYAQEBQCCS
|
8.3 | Ki | 74 | — | |
ZJFCBQXPTQSTCZ
|
8.3 | IC50 | 8 | — | |
RFHIMTLASCGOTR
|
8.3 | IC50 | 3 | — | |
ADFZKKWKESWUFY
|
8.3 | IC50 | 8 | — | |
WOSKHXYHFSIKNG
|
8.3 | IC50 | 24 | — | |
FGPIVIJULBNRBX
|
8.3 | IC50 | 4 | — | |
IDBAAYPNWLPEBC
|
8.2 | IC50 | 2 | — | |
XBBZAHDOGBGKGM
|
8.2 | IC50 | 5 | Yes | |
KUZRTSMZHWGUIV
|
8.2 | IC50 | 2 | — | |
QNDAYXSCYXLLNB
|
8.2 | IC50 | 3 | — | |
FGLRXTXAKOMMOX
|
8.2 | IC50 | 5 | — | |
ONIQOQHATWINJY
|
8.2 | IC50 | 25 | — | |
PKXSPUDURLLHHG
|
8.2 | IC50 | 5 | Yes | |
PUIMLXYJXGFFNV
|
8.2 | IC50 | 4 | — | |
RAHBGWKEPAQNFF
|
8.2 | IC50 | 26 | — | |
WPXVVAWAHQHJPF
|
8.2 | IC50 | 41 | — | |
ADLPKFFMGIJZIM
|
8.2 | Ki | 44 | — | |
FQYLJBVSYHZWLT
|
8.2 | Ki | 35 | Yes | |
HKSZLNNOFSGOKW
|
8.2 | Ki | 118 | — | |
QONPPIZSNSSCSK
|
8.2 | Ki | 45 | Yes | |
XOOAAYRIVATZNM
|
8.2 | Ki | 55 | — | |
GUOKMFDFLUGBPS
|
8.2 | IC50 | 7 | Yes | |
PFPXVMRFOYULPT
|
8.2 | IC50 | 7 | Yes | |
FTERNYMEXWLTAM
|
8.2 | IC50 | 5 | Yes | |
JQDTYPFSLIFJAT
|
8.2 | IC50 | 5 | Yes | |
MOEODMGOTIIAHE
|
8.2 | IC50 | 5 | — | |
PJNSVPCZGALJML
|
8.2 | IC50 | 5 | — | |
DSBPVMDUESDKNK
|
8.1 | IC50 | 9 | Yes | |
KNDPXYAMINMLED
|
8.1 | IC50 | 11 | — | |
ONHZXYNGPZWHBN
|
8.1 | IC50 | 3 | — | |
BFZLDRFGXXMKES
|
8.1 | IC50 | 5 | Yes | |
JZCWLJDSIRUGIN
|
8.1 | Ki | 16 | — | |
KQVFLNYZDGJFNM
|
8.1 | IC50 | 5 | Yes | |
MVJMMLFMPWITEJ
|
8.1 | Ki | 110 | — | |
NRZYTPAJGVTKIM
|
8.1 | Ki | 38 | — | |
TWYCZJMOEMMCGC
|
8.1 | IC50 | 6 | Yes | |
UTQPKPHUIMHAAN
|
8.1 | Ki | 22 | — | |
GGJRNPWQYMGFOS
|
8.1 | IC50 | 2 | — | |
QNSYKQNSCIEOLI
|
8.1 | IC50 | 5 | Yes |