Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSBZFFNSBMBYQA
|
8.7 | IC50 | 9 | — | |
WUBFAXNVDMCVIO
|
8.7 | IC50 | 12 | Yes | |
NMMQJLYMIJYIAK
|
8.7 | IC50 | 3 | — | |
JOAFWIHZEBKYQK
|
8.7 | IC50 | 10 | — | |
OSPKANQURMXUIE
|
8.7 | IC50 | 7 | Yes | |
PLKAJXMYXBXIGX
|
8.7 | IC50 | 7 | Yes | |
ZAJKUNDNLWGYKD
|
8.6 | IC50 | 3 | — | |
UGEJLCNSVIVALC
|
8.6 | Ki | 41 | — | |
SUXYGJZMCWKJJI
|
8.6 | IC50 | 26 | Yes | |
SQQOETQMUXTTJU
|
8.6 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
8.6 | IC50 | 154 | — | |
HCAUEIOBSYOQPN
|
8.5 | IC50 | 5 | Yes | |
IFUCZPASJWTYRU
|
8.5 | IC50 | 5 | — | |
JBJZIAHKSVQDAN
|
8.5 | IC50 | 5 | Yes | |
JPKSISIJPSXDLA
|
8.5 | IC50 | 10 | Yes | |
SPMVMDHWKHCIDT
|
8.5 | IC50 | 30 | — | |
GCYXEGSPUDSZJY
|
8.5 | Ki | 82 | — | |
GDEJPGKNPRJNGE
|
8.5 | Ki | 6 | — | |
GSXRCPJTNIGKSZ
|
8.5 | Ki | 43 | — | |
NSKFXNDKPCVDIN
|
8.5 | Ki | 12 | — | |
RBXYGQNZRVPDNB
|
8.5 | Ki | 34 | — | |
RKLGMDOZEOTQEM
|
8.5 | Ki | 12 | — | |
UOOZSMNSBYVUGZ
|
8.5 | Ki | 32 | — | |
WPHKIQPVPYJNAX
|
8.5 | Ki | 81 | — | |
XHCPCYVQXFHJAU
|
8.5 | IC50 | 12 | — | |
HKSZLNNOFSGOKW
|
8.5 | IC50 | 408 | — | |
SOXNNGFGYDFPDL
|
8.5 | IC50 | 3 | — | |
ZFHLKLQIDSNDHN
|
8.5 | IC50 | 3 | — | |
DTHSJRSUDUUQFI
|
8.4 | IC50 | 3 | — | |
QAGLJDWYCCJEHH
|
8.4 | IC50 | 7 | Yes | |
XXJWYDDUDKYVKI
|
8.4 | IC50 | 52 | — | |
GZQZGOLXVRSKEE
|
8.4 | IC50 | 2 | — | |
AMHUBFWCCMLLCJ
|
8.4 | IC50 | 15 | — | |
BRKGRQVBHFZISR
|
8.4 | IC50 | 7 | Yes | |
FGSVLADZCDNNOC
|
8.4 | Ki | 11 | — | |
FKFACVZGGDYEHZ
|
8.4 | IC50 | 5 | Yes | |
GEGCXGMFUYJULA
|
8.4 | Ki | 30 | Yes | |
LGHBDVLAHHANMX
|
8.4 | Ki | 53 | — | |
MLIFNJABMANKEU
|
8.4 | IC50 | 9 | Yes | |
NRGYZNJPCGRCLV
|
8.4 | Ki | 52 | — | |
QFCXANHHBCGMAS
|
8.4 | IC50 | 7 | — | |
UCSSQROSBFPVKH
|
8.4 | IC50 | 7 | Yes | |
UVNBMNWTGOQKQF
|
8.4 | IC50 | 8 | Yes | |
XJSFDMGICAWQFS
|
8.4 | Ki | 60 | — | |
XKZINYYXWJEYEL
|
8.4 | Ki | 37 | — | |
ZMZOKLZTXMCMNW
|
8.4 | IC50 | 4 | — | |
HPTVZCOLBBFDMI
|
8.4 | IC50 | 3 | — | |
UVZNMKLHIOHOBN
|
8.4 | IC50 | 3 | — | |
UDVJBRYBBSVDDS
|
8.3 | IC50 | 14 | — | |
SPMVMDHWKHCIDT
|
8.3 | IC50 | 5 | — |