Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJZDECGDCKOHBV
|
6.3 | Ki | 70 | — | |
UXMNYFJHEBEDJS
|
6.3 | Ki | 19 | Yes | |
WYOMXSAYYXBPMN
|
6.3 | Ki | 24 | — | |
XGMWRIIMIJPGBH
|
6.3 | Ki | 10 | — | |
YGEACCLUBSGMMJ
|
6.3 | Ki | 16 | — | |
NQHMMDRPRXVCLT
|
6.3 | IC50 | 8 | Yes | |
QTMASMKMHNYBIC
|
6.3 | IC50 | 8 | Yes | |
TXHQSKPOVJIXCS
|
6.3 | IC50 | 3 | — | |
WDZVJGNTRLDPPZ
|
6.3 | IC50 | 3 | — | |
AWJVIOYPZZZYAX
|
6.3 | IC50 | 2 | — | |
FVPYEAORCOKOLV
|
6.3 | IC50 | 6 | — | |
XRUQJEMSXNFQSL
|
6.2 | IC50 | 3 | — | |
HTZHPXKKPOLGTR
|
6.2 | IC50 | 9 | — | |
BHSUCGLRVZHATB
|
6.2 | IC50 | 3 | — | |
UGVYZLLHULWGLZ
|
6.2 | IC50 | 4 | Yes | |
NRNLMJPRICXHLO
|
6.2 | IC50 | 3 | — | |
ZBVKQIOFSQFJCD
|
6.2 | IC50 | 3 | — | |
ZLISHOMLHVNDJG
|
6.2 | IC50 | 3 | — | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
GMFXLDJYMOMKKL
|
6.2 | IC50 | 3 | — | |
GQGMUKOYILWOIQ
|
6.2 | Ki | 25 | — | |
MFMXAWQGPQXDRJ
|
6.2 | Ki | 27 | — | |
PYXQMJSGJIJHJT
|
6.2 | Ki | 28 | — | |
UWQBVYXTLXNIOO
|
6.2 | Ki | 10 | — | |
VXNUSJMWECFYQW
|
6.2 | IC50 | 3 | — | |
ZHTVWJDQZBBZHV
|
6.2 | Ki | 9 | — | |
ZVPDNRVYHLRXLX
|
6.2 | Ki | 35 | Yes | |
LBKSEXFJQLMCIG
|
6.2 | IC50 | 3 | — | |
UFKLYTOEMRFKAD
|
6.2 | IC50 | 6 | — | |
RNIJHXFMJVFHLF
|
6.2 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 91 | Yes | |
UAKYYEQJRKJUBT
|
6.2 | Ki | 5 | Yes | |
GUBJNPWVIUFSTR
|
6.2 | Kd | 103 | — | |
VNDWQCSOSCCWIP
|
6.2 | IC50 | 39 | Yes | |
JWTUFAOHKVRJNA
|
6.1 | IC50 | 5 | Yes | |
JWTUFAOHKVRJNA
|
6.1 | IC50 | 4 | — | |
VAARYSWULJUGST
|
6.1 | Kd | 119 | Yes | |
WCFROKQUHQFBGC
|
6.1 | IC50 | 3 | — | |
AAYZTFLAQXDFOL
|
6.1 | Ki | 11 | — | |
BCNMJLRKWYKBBZ
|
6.1 | IC50 | 4 | — | |
GHMRUNOHAHJNNA
|
6.1 | Ki | 29 | — | |
HHSVICUMCOBRPT
|
6.1 | Ki | 33 | — | |
MTCHQDWUHQADSY
|
6.1 | Ki | 29 | — | |
NHFDRBXTEDBWCZ
|
6.1 | Ki | 41 | — | |
PEXKNSGOEOREKM
|
6.1 | Ki | 13 | — | |
TXHOCWWJSGCZLC
|
6.1 | Ki | 18 | — | |
ULVWJFBHQIXEPE
|
6.1 | Ki | 10 | — | |
UPITUWGOTMBQLX
|
6.1 | Ki | 13 | — | |
WUBHCQHBUVGGRX
|
6.1 | Ki | 11 | — |