Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FYOYABXHBTZQMB
|
6.5 | IC50 | 3 | — | |
HEIWGGHLGABSLB
|
6.5 | Kd | 10 | — | |
SSHDKAJDJAVHAF
|
6.5 | IC50 | 8 | Yes | |
HFGMJNUBHMDODU
|
6.5 | IC50 | 3 | — | |
VKLQCYYJIRWXHJ
|
6.5 | IC50 | 3 | — | |
WWGQYMKITSMXKY
|
6.5 | IC50 | 3 | — | |
ZEXJBANGHOAHDZ
|
6.5 | IC50 | 8 | Yes | |
QCKKTDVCCCBGDD
|
6.5 | IC50 | 8 | — | |
DZNRLDJRJXFYKU
|
6.4 | IC50 | 3 | — | |
ULTCRVJUAZCGPP
|
6.4 | IC50 | 5 | — | |
HTIZPBXCJPQDEM
|
6.4 | IC50 | 4 | Yes | |
GIODDBAYPWNJIQ
|
6.4 | IC50 | 4 | — | |
HBWLNACPIFKNIP
|
6.4 | IC50 | 3 | — | |
SHPFDGWALWEPGS
|
6.4 | Kd | 35 | — | |
DBXGGXLBTWZXBB
|
6.4 | Ki | 39 | — | |
DSBLOQJREHHYBA
|
6.4 | IC50 | 3 | — | |
GDYZFFBMSBDTAA
|
6.4 | Ki | 60 | — | |
NXNQLECPAXXYTR
|
6.4 | Ki | 29 | — | |
PJSBFZAYJQMORO
|
6.4 | Ki | 11 | — | |
PNKALLUVKOKYHZ
|
6.4 | Ki | 32 | — | |
QNUKRWAIZMBVCU
|
6.4 | Ki | 46 | — | |
QQUXFYAWXPMDOE
|
6.4 | Ki | 31 | — | |
RIUZPIBUSOHUKF
|
6.4 | Ki | 23 | — | |
RQJIDUOCLNMUHR
|
6.4 | Ki | 15 | — | |
WVFWTUJEHMVUBG
|
6.4 | Ki | 25 | — | |
XPPLYAKZGXYPOZ
|
6.4 | Ki | 6 | — | |
AIKSEDMIHLRPPQ
|
6.4 | IC50 | 3 | — | |
DGHDMQLWTPPVOS
|
6.4 | IC50 | 3 | — | |
PUIXMSRTTHLNKI
|
6.4 | IC50 | 12 | — | |
CGWDFIYFJPIFIK
|
6.4 | IC50 | 3 | — | |
CKYLEUNHWFIYOR
|
6.4 | IC50 | 3 | — | |
MLLQJNIKDWEEFT
|
6.4 | IC50 | 6 | — | |
XLSPYLMTRXPYKY
|
6.4 | IC50 | 13 | — | |
ZECOHPFWGOCWLO
|
6.4 | IC50 | 5 | — | |
MPASHPJAIUOWCK
|
6.4 | IC50 | 9 | — | |
WNZYDSHFADUYSA
|
6.4 | IC50 | 3 | — | |
AAKJLRGGTJKAMG
|
6.3 | IC50 | 50 | Yes | |
ASBBRVILAUZLPW
|
6.3 | IC50 | 3 | — | |
OTLBXDXENSMYGU
|
6.3 | IC50 | 2 | — | |
SRNHAKVSFVSSPN
|
6.3 | IC50 | 8 | Yes | |
FQGHYVHLTQUXGX
|
6.3 | IC50 | 4 | — | |
JABBQOPTTSFZHZ
|
6.3 | IC50 | 3 | — | |
ARVPXHGQLZVIJF
|
6.3 | IC50 | 3 | — | |
DCYHJVFMNYSPNT
|
6.3 | IC50 | 9 | — | |
DIZVEEIWWJAIEW
|
6.3 | IC50 | 4 | — | |
HEKAIDKUDLCBRU
|
6.3 | Ki | 20 | — | |
HHFBDROWDBDFBR
|
6.3 | Ki | 40 | Yes | |
JVCNXAORTVNADE
|
6.3 | IC50 | 3 | — | |
KWSZYBNXNYRQCC
|
6.3 | Ki | 21 | — | |
NHEQNFWGPSKRMJ
|
6.3 | Ki | 7 | — |