Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RKLRBLPEQCNXFE
|
6.7 | IC50 | 5 | — | |
RYAVJHIPOWNWDE
|
6.7 | Ki | 38 | — | |
ZGZVRPRSFXRGCF
|
6.7 | Ki | 76 | — | |
NOUVYWRJTCFRGO
|
6.7 | IC50 | 2 | — | |
HUJQPYATBOSOGN
|
6.7 | IC50 | 3 | — | |
OVTHZKRCTBBAOW
|
6.7 | IC50 | 5 | Yes | |
QYKZROZZKQVCOO
|
6.7 | IC50 | 3 | — | |
ZUXFIRWLAQBCCS
|
6.7 | IC50 | 8 | Yes | |
VYWXBPWMVHMUQW
|
6.7 | IC50 | 7 | — | |
KRHJQHMWPVTYCU
|
6.6 | IC50 | 6 | — | |
HJFDTNBKNJFDQP
|
6.6 | IC50 | 3 | — | |
UHTHHESEBZOYNR
|
6.6 | IC50 | 66 | Yes | |
DIOWOEJYLCJCNO
|
6.6 | IC50 | 3 | — | |
KAVPZFNKRGDVLL
|
6.6 | IC50 | 2 | — | |
MFAQYJIYDMLAIM
|
6.6 | Kd | 130 | Yes | |
WBQXIIJDZSUXJV
|
6.6 | IC50 | 3 | — | |
WVXNSAVVKYZVOE
|
6.6 | IC50 | 92 | — | |
APUCFXHENVUXCY
|
6.6 | Ki | 15 | — | |
BQWBZBFRJHWSEA
|
6.6 | IC50 | 5 | — | |
CLEGDJQQHUTCOW
|
6.6 | Ki | 43 | — | |
DOLVPVSWTLFZMQ
|
6.6 | Ki | 17 | — | |
GALVWTFFXPRMQM
|
6.6 | Ki | 20 | — | |
IOBVCHJTLVPPBR
|
6.6 | Ki | 39 | — | |
MXAVKSDRMSOCKE
|
6.6 | IC50 | 3 | — | |
MZDKLVOWGIOKTN
|
6.6 | Ki | 80 | — | |
NTPDQTIWAODSAB
|
6.6 | IC50 | 3 | — | |
PCQMERRARZKTPW
|
6.6 | Ki | 68 | — | |
QAWSAMDJZZDGDW
|
6.6 | IC50 | 4 | — | |
QXRJBJVCBQSLTA
|
6.6 | Ki | 29 | — | |
QQOJRBANIUPIQJ
|
6.6 | IC50 | 3 | — | |
KOJNZGHIASJHCV
|
6.6 | IC50 | 3 | — | |
MVCOAUNKQVWQHZ
|
6.6 | IC50 | 54 | Yes | |
RIJLVEAXPNLDTC
|
6.6 | IC50 | 7 | — | |
UAFDWTTZIJTWGE
|
6.6 | IC50 | 2 | — | |
RDWQPGCGRCTSIN
|
6.5 | IC50 | 5 | Yes | |
SADVQUINRBCGFP
|
6.5 | IC50 | 7 | — | |
ODGMIRDHEZREOW
|
6.5 | IC50 | 3 | — | |
ACPOUJIDANTYHO
|
6.5 | IC50 | 17 | Yes | |
DVZRCIHWWHNWKI
|
6.5 | IC50 | 3 | — | |
QKSJQFXYMMEPRF
|
6.5 | IC50 | 3 | — | |
SNEWXKIDJFOZMO
|
6.5 | IC50 | 3 | — | |
WOSBEBRTYHKLTR
|
6.5 | IC50 | 4 | — | |
ACNCCUVYXQGPKZ
|
6.5 | Ki | 31 | — | |
BTHLNBWTKKAULX
|
6.5 | Ki | 16 | — | |
GQLWKGVBOIYMTN
|
6.5 | Ki | 35 | — | |
OAVGBZOFDPFGPJ
|
6.5 | Ki | 42 | Yes | |
PUPCRRRSBUYJAD
|
6.5 | Ki | 44 | Yes | |
RLYVBHARZJDPAR
|
6.5 | IC50 | 3 | — | |
WUWDLXZGHZSWQZ
|
6.5 | Ki | 41 | — | |
ZAARMHXLYCHRAK
|
6.5 | Ki | 20 | — |