Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JPTQVDRPKXSDDN
|
10.0 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
10.0 | IC50 | 43 | — | |
LYHDXABKNJMNEZ
|
9.9 | Ki | 10 | — | |
SXKJHBJVKCAXFA
|
9.7 | IC50 | 3 | — | |
XPVAPOBXNPDLHJ
|
9.7 | IC50 | 3 | — | |
UUVMNPKFPGJBNX
|
9.7 | Ki | 10 | — | |
VPDYUDURNXPNMA
|
9.7 | IC50 | 5 | Yes | |
BDPBZUHWAVABDM
|
9.5 | Ki | 11 | — | |
FOONBYIHFUMRSX
|
9.5 | Ki | 12 | — | |
SJMFZIGFOIPNPE
|
9.5 | Ki | 10 | — | |
WEMHHXYZAJVSME
|
9.5 | IC50 | 3 | — | |
MEBWIBLSBZGQSC
|
9.4 | IC50 | 3 | — | |
NKKLZQAIJJQHIF
|
9.4 | IC50 | 3 | — | |
HQPNLIKXAPLWBQ
|
9.4 | Ki | 12 | Yes | |
JGFZPZGREYNUPH
|
9.4 | IC50 | 5 | Yes | |
ZQQVWTACALNOAJ
|
9.4 | Ki | 11 | — | |
CQGCMAIBZGXOAJ
|
9.4 | IC50 | 3 | — | |
AMRDEKYBJXNLRC
|
9.4 | IC50 | 3 | — | |
NEQZWEXWOFPKOT
|
9.3 | IC50 | 9 | Yes | |
PMCATQTXBPQRSD
|
9.3 | IC50 | 3 | — | |
QEXZHTIPIXJKTN
|
9.2 | IC50 | 3 | — | |
ZFFOQWCQWWHTIS
|
9.2 | IC50 | 3 | — | |
DMTDZFGYURLLKX
|
9.1 | Ki | 13 | Yes | |
MZZIULFUXGVMGF
|
9.1 | IC50 | 3 | — | |
QDOBTYVGPGFRCM
|
9.1 | Ki | 11 | — | |
VMAAFUOXTWPYRN
|
9.1 | IC50 | 9 | Yes | |
YEPNVBNYCRGZRX
|
9.1 | Ki | 26 | — | |
XWFXAJNJXGILIN
|
9.1 | IC50 | 3 | — | |
QXPNJMHRUZCEAP
|
9.0 | IC50 | 14 | — | |
DBXOMQJZSQLQED
|
9.0 | Ki | 12 | — | |
IALDYVNFZAPNJV
|
9.0 | IC50 | 11 | — | |
LOLPPWBBNUVNQZ
|
9.0 | IC50 | 97 | Yes | |
QAKMQVCMEPKBHL
|
9.0 | Ki | 11 | — | |
TTZSNFLLYPYKIL
|
9.0 | IC50 | 7 | — | |
VZRLBUJXKJBRFA
|
9.0 | IC50 | 3 | — | |
DZFZXPPHBWCXPQ
|
9.0 | IC50 | 12 | — | |
OSZVHJYNXBUVAH
|
9.0 | IC50 | 12 | — | |
STINDBVFOPRZHE
|
9.0 | IC50 | 8 | Yes | |
VEVUBFZLKUNGER
|
9.0 | IC50 | 5 | — | |
DELFTXSEBVUJAK
|
8.9 | IC50 | 3 | — | |
PFMPOBVAYMTUOX
|
8.9 | IC50 | 3 | — | |
ZDMGPVTVMCERRZ
|
8.9 | IC50 | 3 | — | |
LKWJIINNTXDWNN
|
8.9 | IC50 | 3 | — | |
KGSRYTUWXUESJK
|
8.9 | IC50 | 7 | — | |
SEJGTFPOEJWEGG
|
8.8 | Kd | 149 | — | |
KROLCVQARUUHNV
|
8.8 | Ki | 12 | — | |
RPDVCUCXMGWTFA
|
8.8 | Ki | 10 | — | |
WJZSUSVUKVZGLF
|
8.7 | IC50 | 7 | Yes | |
DLPARMNJOHFOLU
|
8.7 | Ki | 14 | Yes | |
KSIYIAJUQCMDOR
|
8.7 | IC50 | 2 | — |