Target Details
| UniProt AC | P35626 |
|---|---|
| Gene Symbol | GRK3 |
| Protein Name | G protein-coupled receptor kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 35
- Clinical molecules 1
- Avg pChEMBL 7.11
KEGG Pathways (6)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DMNINFHJFPFPIZ
|
9.2 | IC50 | 4 | — | |
XWJOKKXDMHSILW
|
8.7 | IC50 | 3 | — | |
ARSZMAAOVNYKQN
|
8.5 | IC50 | 3 | — | |
WGESQHUBLPGDDK
|
8.4 | IC50 | 3 | — | |
WFOVEDJTASPCIR
|
8.3 | IC50 | 2 | — | |
FENQBUSSSWWVGH
|
8.0 | Ki | 3 | — | |
LHAZDFBNDIQNSG
|
8.0 | Ki | 4 | — | |
SKZTUPIPRLPDKY
|
8.0 | Ki | 3 | — | |
VRKITNLDCQGIJI
|
8.0 | Ki | 3 | — | |
XHFJYOGNWBJZAX
|
8.0 | Ki | 2 | — | |
MSYSXAOSMCNJKL
|
7.7 | IC50 | 3 | — | |
XYUFCXJZFZPEJD
|
7.3 | IC50 | 23 | Yes | |
BXMIHYGPXLIJBT
|
7.0 | Ki | 2 | — | |
DCJIPWKGABWYAG
|
7.0 | Ki | 2 | — | |
HDOAZITZHWAPBC
|
7.0 | Ki | 2 | — | |
KYWXYKMZNMJBMK
|
7.0 | Ki | 2 | — | |
NDSSSMYGJDDEPB
|
7.0 | Ki | 3 | — | |
PDXVRCZNPFLZJP
|
7.0 | Ki | 3 | — | |
PWMGIYOLYSEHBN
|
7.0 | Ki | 3 | — | |
QNWKTVKWUCLLKW
|
7.0 | Ki | 2 | — | |
RPBKUXXUYPWIPS
|
7.0 | Ki | 3 | — | |
VFKYFTQIVJAIAA
|
7.0 | Ki | 2 | — | |
YKLNVZIGQDKBKJ
|
7.0 | Ki | 3 | — | |
ZXYUSNLUAQYJFK
|
7.0 | Ki | 3 | — | |
RAXZSEGXMBWYQK
|
6.8 | Kd | 21 | — | |
HKSZLNNOFSGOKW
|
6.1 | IC50 | 408 | — | |
CWUZHXXAZSEESR
|
6.0 | Ki | 3 | — | |
GKLCWXCSSBEZOG
|
6.0 | Ki | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KWGIZLMNJXFPFV
|
6.0 | Ki | 3 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
QDNSHFHBLOTJEL
|
6.0 | Ki | 3 | — | |
SGPKBJQYKUQGKV
|
6.0 | Ki | 3 | — | |
XMRRJWMAVDAELT
|
6.0 | Ki | 2 | — |