Target Details
| UniProt AC | P35590 |
|---|---|
| Gene Symbol | TIE1 |
| Protein Name | Tyrosine-protein kinase receptor Tie-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 31
- Clinical molecules 14
- Avg pChEMBL 7.11
Associated Diseases (1)
Active Molecules (31)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODPGGGTTYSGTGO
|
9.5 | Kd | 153 | — | |
QBRQTJMZEYORSP
|
9.1 | Kd | 12 | — | |
CXQHYVUVSFXTMY
|
9.1 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
9.1 | Kd | 149 | — | |
MPASHPJAIUOWCK
|
9.1 | Kd | 9 | — | |
MVCOAUNKQVWQHZ
|
8.1 | Kd | 54 | Yes | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
JSAQBOQCZJHWMA
|
7.4 | Kd | 11 | — | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 213 | — | |
MLDQJTXFUGDVEO
|
7.2 | Kd | 85 | Yes | |
NHHQJBCNYHBUSI
|
7.1 | Kd | 220 | — | |
RITAVMQDGBJQJZ
|
7.0 | Kd | 43 | — | |
KTEIFNKAUNYNJU
|
7.0 | Kd | 114 | — | |
MPVGZUGXCQEXTM
|
7.0 | Kd | 61 | Yes | |
MOONEVNPHKFNGV
|
6.9 | IC50 | 4 | — | |
YABJJWZLRMPFSI
|
6.8 | Kd | 34 | — | |
KDKUVYLMPJIGKA
|
6.6 | Kd | 91 | Yes | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
XXJWYDDUDKYVKI
|
6.5 | Kd | 52 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
QYZOGCMHVIGURT
|
6.5 | Kd | 26 | Yes | |
JWNPDZNEKVCWMY
|
6.4 | Kd | 57 | Yes | |
LQVXSNNAFNGRAH
|
6.2 | Kd | 33 | Yes | |
UIARLYUEJFELEN
|
6.2 | Kd | 289 | Yes | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
CUIHSIWYWATEQL
|
6.2 | Kd | 61 | Yes | |
ZHOXAGNPCZTRBN
|
6.1 | Kd | 20 | — | |
AAKJLRGGTJKAMG
|
6.1 | Kd | 50 | Yes | |
HHZIURLSWUIHRB
|
6.0 | Kd | 57 | Yes | |
WVUNYSQLFKLYNI
|
6.0 | Kd | 46 | Yes |