Target Details
| UniProt AC | P35499 |
|---|---|
| Gene Symbol | SCN4A |
| Protein Name | Sodium channel protein type 4 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) |
Summary
- Multi-target molecules 99
- Clinical molecules 0
- Avg pChEMBL 6.81
Associated Diseases (8)
Active Molecules (99)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVQFYGIEBVVYRN
|
6.7 | IC50 | 4 | — | |
RCPXNDYGDIWIIH
|
6.7 | IC50 | 2 | — | |
LKNQEIFVYZPGTP
|
6.6 | IC50 | 2 | — | |
RSVKRFJKRDUBHP
|
6.6 | IC50 | 2 | — | |
SGQSMRQYEPPNIA
|
6.6 | Ki | 2 | — | |
VBPFCFPZENVMHX
|
6.6 | IC50 | 2 | — | |
IVVQUXZDEFTOMS
|
6.6 | IC50 | 2 | — | |
MOGUMJAJYFSRJV
|
6.6 | IC50 | 3 | — | |
TWMQZRRRRZWVGV
|
6.5 | IC50 | 2 | — | |
LONCXOHJDPUEJD
|
6.5 | IC50 | 2 | — | |
XYQBMTXAQVNHCL
|
6.5 | IC50 | 2 | — | |
ZJNBTZRRUMSOPS
|
6.4 | IC50 | 2 | — | |
QLKAFHZJICDACE
|
6.4 | IC50 | 3 | — | |
REZDHPKOVBPAMP
|
6.4 | IC50 | 2 | — | |
VYGMELUEYAGXCD
|
6.4 | IC50 | 2 | — | |
AYYNSJQIJFSWRU
|
6.4 | IC50 | 2 | — | |
DCMQCUNWFWGVDN
|
6.4 | IC50 | 2 | — | |
DMXSSTRXUNIILQ
|
6.3 | IC50 | 2 | — | |
IPRFOFLOYPAGPA
|
6.3 | IC50 | 2 | — | |
IXXSLXXUOAYZEZ
|
6.3 | IC50 | 2 | — | |
ZDYIMJLPMWNRHT
|
6.3 | IC50 | 2 | — | |
VWANWFMHXJKMFY
|
6.3 | IC50 | 2 | — | |
LBUJARQQUVGRHC
|
6.3 | IC50 | 2 | — | |
FYISQNWWCJCJBP
|
6.3 | IC50 | 2 | — | |
MHEJDCLHINDVMO
|
6.2 | IC50 | 2 | — | |
OEDXJWJKZWZZTK
|
6.2 | IC50 | 2 | — | |
XJXFPLHCRFQLST
|
6.2 | IC50 | 3 | — | |
YYGZVYTVCWHOFB
|
6.2 | IC50 | 2 | — | |
OGZOWARNWAFKNY
|
6.2 | IC50 | 2 | — | |
OGZOWARNWAFKNY
|
6.2 | IC50 | 2 | — | |
DXOIDXNPYTZMEK
|
6.2 | IC50 | 2 | — | |
ISXFEVUJMHDJDV
|
6.2 | IC50 | 2 | — | |
NNJOTOMAUDKXKD
|
6.2 | IC50 | 2 | — | |
UGOYONMBZFCBPL
|
6.2 | IC50 | 2 | — | |
XWNXLYNIWAXGBY
|
6.2 | IC50 | 2 | — | |
XYPMZYYZUJQOOS
|
6.2 | IC50 | 2 | — | |
MIOZPPVHYXVEIY
|
6.1 | IC50 | 2 | — | |
VGHUQOPCSXOUJD
|
6.1 | IC50 | 2 | — | |
MLPXAEWHSAPBSG
|
6.1 | IC50 | 2 | — | |
BENAISSLCJROOE
|
6.1 | IC50 | 2 | — | |
KQMXRQQDPACMRM
|
6.1 | IC50 | 2 | — | |
JKTHEHVHKZOFOB
|
6.1 | IC50 | 2 | — | |
FOXHBDLHQXLGGN
|
6.0 | IC50 | 2 | — | |
IFOFQYZJHRNQLW
|
6.0 | IC50 | 2 | — | |
VDZFYIRHQIKGSV
|
6.0 | IC50 | 2 | — | |
YFPFSPWJNLLSJF
|
6.0 | IC50 | 2 | — | |
YFRDMCXBZDPRIB
|
6.0 | IC50 | 2 | — | |
HBNPJJILLOYFJU
|
6.0 | IC50 | 21 | — | |
VGRYEIIRDYDLIT
|
6.0 | IC50 | 2 | — |