Target Details
| UniProt AC | P35499 |
|---|---|
| Gene Symbol | SCN4A |
| Protein Name | Sodium channel protein type 4 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) |
Summary
- Multi-target molecules 99
- Clinical molecules 0
- Avg pChEMBL 6.81
Associated Diseases (8)
Active Molecules (99)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BJJIKPMJNDTIHW
|
10.2 | IC50 | 3 | — | |
KGGOSMYISLXZHL
|
8.7 | IC50 | 2 | — | |
PIGHRURPFWHXDQ
|
8.7 | IC50 | 2 | — | |
SXOAHIZWCZOILH
|
8.5 | IC50 | 9 | — | |
CFMYXEVWODSLAX
|
8.1 | IC50 | 8 | — | |
PTCBNPULJWGSML
|
8.1 | IC50 | 9 | — | |
ZQXXVCXFDRFOAC
|
7.8 | IC50 | 2 | — | |
RPQXVSUAYFXFJA
|
7.7 | IC50 | 8 | — | |
JMMCZELYPMWMKB
|
7.7 | IC50 | 2 | — | |
RBQRPVYHDUYUMZ
|
7.7 | IC50 | 2 | — | |
AHWSGUQUIABDFY
|
7.6 | IC50 | 2 | — | |
LRYGMRYJDQOKLI
|
7.6 | IC50 | 2 | — | |
KYBPOTYVFWNSGS
|
7.5 | Kd | 8 | — | |
VRRIYZJUSNMZMP
|
7.5 | IC50 | 2 | — | |
HLJJNNPHQAQLII
|
7.5 | IC50 | 2 | — | |
DFFVMIVCNSUZRH
|
7.4 | IC50 | 2 | — | |
GPPTZPCHCLOBIL
|
7.4 | IC50 | 2 | — | |
KQQXPTRMUYKUIC
|
7.3 | Kd | 8 | — | |
XOAUGYVLRSCGBG
|
7.3 | IC50 | 8 | — | |
JASALYCADJWQID
|
7.3 | IC50 | 2 | — | |
QGQKYSJJEUMYCP
|
7.3 | IC50 | 2 | — | |
VEEQSZWXUOUXPZ
|
7.3 | IC50 | 5 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
GRYVZXPJYFDBIS
|
7.2 | IC50 | 2 | — | |
LZJKVSDOJZQQKC
|
7.1 | IC50 | 2 | — | |
LPJFOYUXGSRSAK
|
7.1 | IC50 | 2 | — | |
NNBQSDGKUCGYMG
|
7.0 | IC50 | 2 | — | |
ZRPWGKPPPKBYAL
|
7.0 | IC50 | 2 | — | |
PTMJZFRCKPOPSW
|
7.0 | IC50 | 2 | — | |
VRUSWBLOISBSSJ
|
7.0 | IC50 | 5 | — | |
BBSAEKOKKBAQRH
|
7.0 | IC50 | 2 | — | |
LXWQXQGRQCXLOL
|
7.0 | IC50 | 2 | — | |
WGQMMWFPSAVNAJ
|
7.0 | IC50 | 2 | — | |
SUDPJHWRLKPICV
|
7.0 | IC50 | 3 | — | |
JYYKEMPXQHPLKT
|
7.0 | IC50 | 3 | — | |
LLCJMXUOUAGOJT
|
6.9 | IC50 | 3 | — | |
PEIYHGIZJQATLS
|
6.9 | IC50 | 2 | — | |
ZUPILDXMDFYYGB
|
6.9 | IC50 | 2 | — | |
DFBDAHMZXJYZJG
|
6.8 | IC50 | 7 | — | |
NLDXBSUTMUSGMG
|
6.8 | IC50 | 2 | — | |
AAUMZZJEGXJINE
|
6.8 | IC50 | 3 | — | |
XINCOPAGFDEGQZ
|
6.8 | IC50 | 2 | — | |
WWSWLMWIXLNWHP
|
6.8 | IC50 | 2 | — | |
MHUUDVZSPFRUSK
|
6.8 | Ki | 2 | — | |
QEITUNTXHQTCMZ
|
6.8 | IC50 | 2 | — | |
KIIZVCWLLOZRPV
|
6.7 | IC50 | 2 | — | |
MHUUDVZSPFRUSK
|
6.7 | Ki | 2 | — | |
BQVSSPNOFJNEHA
|
6.7 | IC50 | 2 | — | |
GUMIVJFWYYSBKF
|
6.7 | IC50 | 2 | — | |
RJKGEAHOEVLLLG
|
6.7 | IC50 | 2 | — |