Target Details
| UniProt AC | P35498 |
|---|---|
| Gene Symbol | SCN1A |
| Protein Name | Sodium channel protein type 1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 542
- Clinical molecules 4
- Avg pChEMBL 7.76
KEGG Pathways (1)
Associated Diseases (6)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HBYPLMPPHBGEDI
|
7.9 | IC50 | 2 | — | |
IRFMFQQIANLALO
|
7.9 | IC50 | 2 | — | |
NEWRVLYCADPFOU
|
7.9 | IC50 | 2 | — | |
PCWUHIYHTMODIL
|
7.9 | IC50 | 2 | — | |
SCZYLEWDHRXONF
|
7.9 | IC50 | 2 | — | |
DUTBELDPUMKBDW
|
7.8 | IC50 | 2 | — | |
GFVCFLPKZWOAQW
|
7.8 | IC50 | 2 | — | |
NZLJRXFUYNPRME
|
7.8 | IC50 | 2 | — | |
PLZANXMHAHDQEY
|
7.8 | IC50 | 2 | — | |
RHLSSDADJRDXLU
|
7.8 | IC50 | 2 | — | |
WHVCUTYOIICUIK
|
7.8 | IC50 | 2 | — | |
ZHOVMQJWRQDRFQ
|
7.8 | IC50 | 2 | — | |
CDWKRWXCVDRSRN
|
7.8 | IC50 | 2 | — | |
GCVLCXXOZKDWKX
|
7.8 | IC50 | 2 | — | |
GIYHIVFXKAMIDY
|
7.8 | IC50 | 2 | — | |
KYERELZTVNAFJL
|
7.8 | IC50 | 2 | — | |
LYTCVQQGCSNFJU
|
7.8 | IC50 | 3 | — | |
OXLXEJBCNSQASQ
|
7.8 | IC50 | 2 | — | |
SJCKDZDWCFXPHT
|
7.8 | IC50 | 2 | — | |
VLIGDXLMKUKWJZ
|
7.8 | IC50 | 2 | — | |
WXFLUTLJETXITM
|
7.8 | IC50 | 2 | — | |
CQOUGURSFKSLMF
|
7.8 | IC50 | 2 | — | |
FNXPIKCUIQCFFD
|
7.8 | IC50 | 2 | — | |
QEQUMUCQZCHHBH
|
7.8 | IC50 | 2 | — | |
QJNYOQCRJJMAOZ
|
7.8 | IC50 | 3 | — | |
XOAUGYVLRSCGBG
|
7.8 | IC50 | 8 | — | |
YJHJXTTXJRZIOQ
|
7.8 | IC50 | 2 | — | |
AUMPIEINVCBDOI
|
7.8 | IC50 | 2 | — | |
GCVLCXXOZKDWKX
|
7.8 | IC50 | 2 | — | |
HBNLKZBNOCBHIO
|
7.8 | IC50 | 2 | — | |
NDHYFBZFYCXQJV
|
7.8 | IC50 | 2 | — | |
OGXYRLBTADEONS
|
7.8 | IC50 | 2 | — | |
VDOLFGHRDHGMCS
|
7.8 | IC50 | 2 | — | |
BJUGCVMDGAASCX
|
7.7 | IC50 | 2 | — | |
VQBGPJJILMRFBJ
|
7.7 | IC50 | 2 | — | |
RAMYNPHHIXANPH
|
7.7 | IC50 | 2 | — | |
YSAHUUYUAWFVKI
|
7.7 | IC50 | 2 | — | |
BJUGCVMDGAASCX
|
7.7 | IC50 | 2 | — | |
DLVHLOHKEQWDBO
|
7.7 | IC50 | 2 | — | |
OVHKFCHMFRAKJC
|
7.7 | IC50 | 2 | — | |
RCAXTKUIFXSBJK
|
7.7 | IC50 | 2 | — | |
SREGSGWKZFYIDY
|
7.7 | IC50 | 3 | — | |
ZUXRUQOEFBOTGF
|
7.7 | IC50 | 4 | — | |
BSHIKYSNYVZEIY
|
7.7 | IC50 | 2 | — | |
CQNROXJZTLLINO
|
7.7 | IC50 | 2 | — | |
HBNLKZBNOCBHIO
|
7.7 | IC50 | 2 | — | |
DLVHLOHKEQWDBO
|
7.7 | IC50 | 2 | — | |
JBECBHNSFAXSII
|
7.7 | IC50 | 2 | — | |
TXWCGOIFALQYHQ
|
7.7 | IC50 | 2 | — | |
UVPFUHLMKQGWHA
|
7.7 | IC50 | 2 | — |