Target Details
| UniProt AC | P35498 |
|---|---|
| Gene Symbol | SCN1A |
| Protein Name | Sodium channel protein type 1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 542
- Clinical molecules 4
- Avg pChEMBL 7.76
KEGG Pathways (1)
Associated Diseases (6)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOTZMAHOBVGVQU
|
8.2 | IC50 | 3 | — | |
DQSHMENCHXKIOD
|
8.2 | IC50 | 2 | — | |
FLRIBHCWDYEBHH
|
8.2 | IC50 | 2 | — | |
GFDXIUXAFNREKM
|
8.2 | IC50 | 6 | — | |
HJRAXXVKFXITKI
|
8.2 | IC50 | 2 | — | |
IKGSSFBIKHWXLY
|
8.2 | IC50 | 2 | — | |
KMXYAYHLGANJIA
|
8.2 | IC50 | 2 | — | |
WFIDFECCLBIDBW
|
8.2 | IC50 | 2 | — | |
ABFJGJYHHOCPJV
|
8.2 | IC50 | 2 | — | |
BRVBRZABHLGTRI
|
8.2 | IC50 | 2 | — | |
GQIRJGCLEQYBML
|
8.2 | IC50 | 3 | — | |
MKTFWIFFQBKEFV
|
8.2 | IC50 | 2 | — | |
NQDCRCJMPKRFBR
|
8.2 | IC50 | 2 | — | |
QJCLEBMUIYIWPM
|
8.2 | IC50 | 2 | — | |
GQIRJGCLEQYBML
|
8.2 | IC50 | 3 | — | |
QIQDHFDWFWPFKT
|
8.2 | IC50 | 2 | — | |
BBTLYGRMWYLRGJ
|
8.2 | IC50 | 2 | — | |
IMNAMBYRWSGKHX
|
8.2 | IC50 | 3 | — | |
LRXJCQGUTGFUKQ
|
8.2 | IC50 | 2 | — | |
VONKMVXDHIRYQE
|
8.2 | IC50 | 2 | — | |
WJLZKECJHILDNE
|
8.2 | IC50 | 2 | — | |
AGUMLPYUAXPZOR
|
8.2 | IC50 | 2 | — | |
YENVCDVPWRTJND
|
8.2 | IC50 | 2 | — | |
QMRDOUTXSQARSD
|
8.2 | IC50 | 2 | — | |
UHSPKNDHOJXKCW
|
8.2 | IC50 | 2 | — | |
VOGXZTHYVIFHTJ
|
8.2 | IC50 | 2 | — | |
HSLPMVWAEHCEIS
|
8.2 | IC50 | 2 | — | |
NSVXLSVOTLNFBX
|
8.2 | IC50 | 2 | — | |
PDJHPFGJNBYHNZ
|
8.2 | IC50 | 2 | — | |
CBIUHBBBOUSNQK
|
8.2 | IC50 | 2 | — | |
VBKZDPSLLFEXQC
|
8.2 | IC50 | 2 | — | |
GPMUUALSFJEQGL
|
8.1 | IC50 | 2 | — | |
OBLNMGFBACQBBP
|
8.1 | IC50 | 2 | — | |
PJGWILKULVRVIE
|
8.1 | IC50 | 2 | — | |
RINFWXVZBUREQN
|
8.1 | IC50 | 2 | — | |
ZHTUHCKSYHDWAK
|
8.1 | IC50 | 2 | — | |
GLJJNWDWTRCSQC
|
8.1 | IC50 | 2 | — | |
MDLDNPVKBYFOTI
|
8.1 | IC50 | 2 | — | |
CQNROXJZTLLINO
|
8.1 | IC50 | 2 | — | |
XFGAFLXHZAYTAU
|
8.1 | IC50 | 2 | — | |
CYBOBMVXTOTJEC
|
8.1 | IC50 | 2 | — | |
DVPUCKCSNKRQIM
|
8.1 | IC50 | 2 | — | |
NSVXLSVOTLNFBX
|
8.1 | IC50 | 2 | — | |
CYBOBMVXTOTJEC
|
8.1 | IC50 | 2 | — | |
LGOHKZMXBAADMN
|
8.1 | IC50 | 2 | — | |
QQSAJPXJGRDAMG
|
8.1 | IC50 | 2 | — | |
GRFFUKNFLUHFHE
|
8.1 | IC50 | 2 | — | |
MARFCZKCASKJQG
|
8.1 | IC50 | 2 | — | |
QMOLJXRAMAPQPQ
|
8.1 | IC50 | 2 | — | |
UHNGVVPJTQLYJP
|
8.1 | IC50 | 2 | — |