Target Details
| UniProt AC | P35498 |
|---|---|
| Gene Symbol | SCN1A |
| Protein Name | Sodium channel protein type 1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 542
- Clinical molecules 4
- Avg pChEMBL 7.76
KEGG Pathways (1)
Associated Diseases (6)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GRFFUKNFLUHFHE
|
8.3 | IC50 | 2 | — | |
QMMKZCBSRMHBGN
|
8.3 | IC50 | 2 | — | |
RJJRKJYXPONNFC
|
8.3 | IC50 | 2 | — | |
AFMUVNRIPITERN
|
8.3 | IC50 | 2 | — | |
APUFQCSYCHYZIW
|
8.3 | IC50 | 2 | — | |
BSGXIJLWDIVEFC
|
8.3 | IC50 | 2 | — | |
CWAAFDMFNOVWLT
|
8.3 | IC50 | 2 | — | |
DEFPDGLJZGBIGF
|
8.3 | IC50 | 2 | — | |
JHWZVZSMRWIZMO
|
8.3 | IC50 | 2 | — | |
CBIUHBBBOUSNQK
|
8.3 | IC50 | 2 | — | |
KBNXSZUPQRGYNY
|
8.3 | IC50 | 3 | — | |
YKHDDBRKQAIROO
|
8.3 | IC50 | 3 | — | |
DHSOPLGHCCWMQK
|
8.3 | IC50 | 3 | — | |
FKPOFESGNHGZMW
|
8.3 | IC50 | 2 | — | |
FKPOFESGNHGZMW
|
8.3 | IC50 | 2 | — | |
KHAPUVAAGNEHQW
|
8.3 | IC50 | 2 | — | |
PRCIGHMFXRYAIG
|
8.3 | IC50 | 3 | — | |
QQRDUMOOLIZBOV
|
8.3 | IC50 | 2 | — | |
RJZUNWGDQAGCHL
|
8.3 | IC50 | 2 | — | |
XDAKREHNKKKEAQ
|
8.3 | IC50 | 2 | — | |
ZVROQFJWLWNYPQ
|
8.3 | IC50 | 2 | — | |
KTQITWVXYXCIPI
|
8.3 | IC50 | 2 | — | |
LKWRNZBTPSCWJT
|
8.3 | IC50 | 3 | — | |
WWPICVXQOKPCAZ
|
8.3 | IC50 | 2 | — | |
YSEGGAVVNUBFOR
|
8.3 | IC50 | 2 | — | |
BHNHPSMLNIXZEA
|
8.3 | IC50 | 2 | — | |
FUFQYXJEKPAYHJ
|
8.3 | IC50 | 2 | — | |
ICDZOMMZQJGZGT
|
8.3 | IC50 | 2 | — | |
LNZNUXVENBAPOZ
|
8.3 | IC50 | 2 | — | |
PBBRTUUYKGXANR
|
8.3 | IC50 | 2 | — | |
QWKZXVRTHGUGEI
|
8.3 | IC50 | 2 | — | |
UUYBPWNOSQSJHQ
|
8.3 | IC50 | 2 | — | |
YEUQOLDVWRDBED
|
8.3 | IC50 | 2 | — | |
ZVROQFJWLWNYPQ
|
8.3 | IC50 | 2 | — | |
BVOXFWHQWQANHR
|
8.3 | IC50 | 2 | — | |
BYPCGZJBGJSUGQ
|
8.3 | IC50 | 2 | — | |
IDJPUZREEMOMJC
|
8.3 | IC50 | 2 | — | |
IKDXHRATCNECAM
|
8.3 | IC50 | 2 | — | |
JEZPXQKQZQRRMC
|
8.3 | IC50 | 2 | — | |
HRRHRSSCWYTCBS
|
8.2 | IC50 | 3 | — | |
IVNAEBIOSDTKSX
|
8.2 | IC50 | 2 | — | |
MQBAFWXBAHSNIS
|
8.2 | IC50 | 2 | — | |
DDOIQOFHDMJGBP
|
8.2 | IC50 | 2 | — | |
DPKBSJIWLASXHR
|
8.2 | IC50 | 2 | — | |
GNHOWCLPSIXZMF
|
8.2 | IC50 | 2 | — | |
HDQYQOWHBKXUCR
|
8.2 | IC50 | 2 | — | |
KRRQPHNWSHNADQ
|
8.2 | IC50 | 2 | — | |
QFOGEZLLIKAJNO
|
8.2 | IC50 | 2 | — | |
VQJZDKCEVLXOTH
|
8.2 | IC50 | 2 | — | |
OCUQANFWZAMQKA
|
8.2 | IC50 | 2 | — |