Target Details
| UniProt AC | P35498 |
|---|---|
| Gene Symbol | SCN1A |
| Protein Name | Sodium channel protein type 1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 542
- Clinical molecules 4
- Avg pChEMBL 7.76
KEGG Pathways (1)
Associated Diseases (6)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YEEDVFRTJANVAV
|
8.5 | IC50 | 2 | — | |
ALEKFWIWCIMWKG
|
8.4 | IC50 | 3 | — | |
ANUDJEBSNITMOR
|
8.4 | IC50 | 2 | — | |
JOYIGLXPDBYYRY
|
8.4 | IC50 | 2 | — | |
LNFPXDBTSWLDMB
|
8.4 | IC50 | 2 | — | |
VCFCDMFIOHFMNG
|
8.4 | IC50 | 2 | — | |
YLPZZUYEMQKXPL
|
8.4 | IC50 | 2 | — | |
ICDZOMMZQJGZGT
|
8.4 | IC50 | 2 | — | |
JZQURVBEWWCEHW
|
8.4 | IC50 | 2 | — | |
WEKXUMJLGXGLNE
|
8.4 | IC50 | 2 | — | |
BGTDJFUYZQLYLF
|
8.4 | IC50 | 2 | — | |
IFEGKGXITIRTCE
|
8.4 | IC50 | 2 | — | |
LHKFTDVGHHDMKX
|
8.4 | IC50 | 2 | — | |
MNTIFTYMXHJTKW
|
8.4 | IC50 | 2 | — | |
REXKPUWAXOQORC
|
8.4 | IC50 | 2 | — | |
UHTDRCGXSYGMRR
|
8.4 | IC50 | 2 | — | |
KBNXSZUPQRGYNY
|
8.4 | IC50 | 2 | — | |
SXOAHIZWCZOILH
|
8.4 | IC50 | 3 | — | |
VCYUDKGDSCTDPU
|
8.4 | IC50 | 2 | — | |
VKRFQEVWFMGEEK
|
8.4 | IC50 | 2 | — | |
XRNKNZSYIMJPQE
|
8.4 | IC50 | 2 | — | |
XRNKNZSYIMJPQE
|
8.4 | IC50 | 2 | — | |
YLPZZUYEMQKXPL
|
8.4 | IC50 | 3 | — | |
AHLGPCZDAPQKRY
|
8.4 | IC50 | 2 | — | |
DDOIQOFHDMJGBP
|
8.4 | IC50 | 2 | — | |
UZDFKZMJYSQQHI
|
8.4 | IC50 | 2 | — | |
VBKZDPSLLFEXQC
|
8.4 | IC50 | 2 | — | |
YGLOZPVIZVIBDT
|
8.4 | IC50 | 2 | — | |
AZHGECCHCQEMBR
|
8.4 | IC50 | 2 | — | |
CFMYXEVWODSLAX
|
8.4 | IC50 | 8 | — | |
ANUDJEBSNITMOR
|
8.4 | IC50 | 2 | — | |
CYVICQCUAYMJDA
|
8.4 | IC50 | 2 | — | |
ICDZOMMZQJGZGT
|
8.4 | IC50 | 2 | — | |
PJGWILKULVRVIE
|
8.4 | IC50 | 2 | — | |
ATFPRZUKXKQMOY
|
8.4 | IC50 | 2 | — | |
MWSVLDOKXAVVNZ
|
8.4 | IC50 | 3 | — | |
SDFWLGIHLRLHLP
|
8.4 | IC50 | 3 | — | |
FCTMRPTVPHVTTN
|
8.4 | IC50 | 3 | — | |
OCNOGKDYKRVBCZ
|
8.4 | IC50 | 3 | — | |
OCUQANFWZAMQKA
|
8.4 | IC50 | 2 | — | |
OZRIMKPTCZSADH
|
8.4 | IC50 | 2 | — | |
SQHCXAPOOMTODU
|
8.4 | IC50 | 2 | — | |
YGLOZPVIZVIBDT
|
8.4 | IC50 | 2 | — | |
GULOFVVKGUTUDX
|
8.3 | IC50 | 2 | — | |
HDCONQSFHGFUFZ
|
8.3 | IC50 | 2 | — | |
KQVZYWXQAVPSNP
|
8.3 | IC50 | 2 | — | |
NDHYFBZFYCXQJV
|
8.3 | IC50 | 2 | — | |
YTJUXLJKPMJRBK
|
8.3 | IC50 | 2 | — | |
CAOWMPQVHUJGPS
|
8.3 | IC50 | 2 | — | |
SAECGYZACNUJAE
|
8.3 | IC50 | 2 | — |