Target Details
| UniProt AC | P35498 |
|---|---|
| Gene Symbol | SCN1A |
| Protein Name | Sodium channel protein type 1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 542
- Clinical molecules 4
- Avg pChEMBL 7.76
KEGG Pathways (1)
Associated Diseases (6)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LJDHLZQUJUBCSY
|
8.6 | IC50 | 2 | — | |
LJOFBQKPPMGKQF
|
8.6 | IC50 | 2 | — | |
SXOAHIZWCZOILH
|
8.6 | IC50 | 2 | — | |
VCFCDMFIOHFMNG
|
8.6 | IC50 | 2 | — | |
VKBNOHOCPXCCEY
|
8.6 | IC50 | 2 | — | |
YJDICZSISKZEKO
|
8.6 | IC50 | 2 | — | |
QZNDZQCKQVDMLB
|
8.6 | IC50 | 2 | — | |
AQQPEEVAXMWVEY
|
8.5 | IC50 | 2 | — | |
DHMIQEWWFKEVEE
|
8.5 | IC50 | 2 | — | |
IZFIUFGSCXTJMM
|
8.5 | IC50 | 2 | — | |
JHTVWHDWWCEEAL
|
8.5 | IC50 | 2 | — | |
PPNSUOZZLIDACH
|
8.5 | IC50 | 2 | — | |
SWJVLLZRHPUGDQ
|
8.5 | IC50 | 2 | — | |
WMAUVGOSBMOBSZ
|
8.5 | IC50 | 2 | — | |
YLOGZZPFMFZBLY
|
8.5 | IC50 | 2 | — | |
YLPZZUYEMQKXPL
|
8.5 | IC50 | 2 | — | |
YYBNTCMQMFIHRU
|
8.5 | IC50 | 2 | — | |
ZYWBKPBGYHQNDP
|
8.5 | IC50 | 2 | — | |
GWODAUIHUKCBIF
|
8.5 | IC50 | 2 | — | |
ABSISAIFUWQGDW
|
8.5 | IC50 | 2 | — | |
AGNWXMAUWNAUTK
|
8.5 | IC50 | 2 | — | |
GNKRHBPEEQTZMU
|
8.5 | IC50 | 2 | — | |
JEQSMTYUSZSZKB
|
8.5 | IC50 | 2 | — | |
KRNHAUPCKRIYSK
|
8.5 | IC50 | 3 | — | |
DEFPDGLJZGBIGF
|
8.5 | IC50 | 2 | — | |
FCGCWVRBOOKMTK
|
8.5 | IC50 | 3 | — | |
KHSJWWIRIZMXGO
|
8.5 | IC50 | 2 | — | |
MFYFOYKTBPOPEW
|
8.5 | IC50 | 2 | — | |
PMHATIGSOAJRQC
|
8.5 | IC50 | 2 | — | |
YMFXBFBMVCEBGO
|
8.5 | IC50 | 2 | — | |
ZJQJBMYDTSMDTO
|
8.5 | IC50 | 2 | — | |
OSHHICZYAPYLTD
|
8.5 | IC50 | 2 | — | |
SJRMDWHBLAJJOP
|
8.5 | IC50 | 2 | — | |
ZZPCDLASCPKEDD
|
8.5 | IC50 | 2 | — | |
AWGKELNBCIVSRF
|
8.5 | IC50 | 2 | — | |
JCGRPZMJTUDYEM
|
8.5 | IC50 | 2 | — | |
JOYIGLXPDBYYRY
|
8.5 | IC50 | 2 | — | |
JZQURVBEWWCEHW
|
8.5 | IC50 | 2 | — | |
UZDFKZMJYSQQHI
|
8.5 | IC50 | 2 | — | |
XBMVGKUHNIZGOK
|
8.5 | IC50 | 2 | — | |
BVXDDXBPDJMLDH
|
8.5 | IC50 | 2 | — | |
FMFYHAKGBTVJEQ
|
8.5 | IC50 | 2 | — | |
FQIILMZKICAGTI
|
8.5 | IC50 | 2 | — | |
PJPZLNSZJCAXGK
|
8.5 | IC50 | 2 | — | |
AOWBBEBBSXNAJF
|
8.5 | IC50 | 2 | — | |
IKDXHRATCNECAM
|
8.5 | IC50 | 2 | — | |
NMBFEULXPSSJAD
|
8.5 | IC50 | 2 | — | |
OHBBONZPZRTSGV
|
8.5 | IC50 | 2 | — | |
QZFIAUDHZFQMKI
|
8.5 | IC50 | 2 | — | |
YEEDVFRTJANVAV
|
8.5 | IC50 | 2 | — |