Target Details
| UniProt AC | P35398 |
|---|---|
| Gene Symbol | RORA |
| Protein Name | Nuclear receptor ROR-alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 37
- Clinical molecules 0
- Avg pChEMBL 6.54
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (37)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OYXZMSRRJOYLLO
|
7.9 | Ki | 2 | — | |
OYXZMSRRJOYLLO
|
7.9 | Ki | 2 | — | |
GIJYGRLHNVZBPZ
|
7.3 | IC50 | 2 | — | |
NOGDJCUSTNXIOS
|
7.2 | IC50 | 2 | — | |
UOLYGIMYNWWJPJ
|
7.2 | IC50 | 3 | — | |
YJGVMLPVUAXIQN
|
7.1 | IC50 | 19 | — | |
XNZJHNCNFWAVAE
|
7.0 | IC50 | 3 | — | |
SGIWFELWJPNFDH
|
6.9 | Ki | 6 | — | |
XGHUJWTXGMRXEL
|
6.9 | IC50 | 3 | — | |
DOVJOUHJSWWBDX
|
6.8 | IC50 | 3 | — | |
OZBSSKGBKHOLGA
|
6.8 | Ki | 2 | — | |
QSMVBOULCKMAMR
|
6.7 | IC50 | 2 | — | |
SHGAZHPCJJPHSC
|
6.7 | IC50 | 13 | — | |
AUVVAXYIELKVAI
|
6.5 | IC50 | 10 | — | |
XEXLJHXWQVDFRD
|
6.5 | IC50 | 2 | — | |
DQKJOHPFSRRCND
|
6.5 | IC50 | 3 | — | |
XHARTEHOSRSMSF
|
6.4 | IC50 | 4 | — | |
CJSMGQLUSXOBBD
|
6.4 | IC50 | 3 | — | |
XRCKIQRUBBOFOL
|
6.4 | IC50 | 2 | — | |
XHJJPQRLFFDDTQ
|
6.4 | IC50 | 5 | — | |
HJJYGXDBXQAVQG
|
6.3 | IC50 | 2 | — | |
PTOAARAWEBMLNO
|
6.2 | IC50 | 3 | — | |
XRLOVVNQWKZVHK
|
6.2 | IC50 | 3 | — | |
NOFOAYPPHIUXJR
|
6.2 | IC50 | 5 | — | |
QQIBJFMXQBDPGQ
|
6.2 | IC50 | 2 | — | |
KGISTBTWGCVWQU
|
6.2 | IC50 | 2 | — | |
ODLLKRFSXYKRQB
|
6.2 | Ki | 2 | — | |
POAKEIXFPDIYHH
|
6.2 | IC50 | 3 | — | |
CHMQQIFPOIZPIJ
|
6.1 | IC50 | 2 | — | |
OTPVLJJKRBOIJC
|
6.1 | IC50 | 2 | — | |
SLGRAIAQIAUZAQ
|
6.1 | IC50 | 16 | — | |
WXQUZMCQBBNKNQ
|
6.1 | IC50 | 2 | — | |
XUFPHJFOAMPPQQ
|
6.1 | IC50 | 2 | — | |
XAVNIJZYVBDIPG
|
6.1 | IC50 | 2 | — | |
JXHFEOAFQXPYIJ
|
6.1 | IC50 | 5 | — | |
NXHAXIRXWHSYTI
|
6.0 | IC50 | 2 | — | |
BKZOIKUBPIWBKV
|
6.0 | IC50 | 3 | — |