Target Details
| UniProt AC | P35372 |
|---|---|
| Gene Symbol | OPRM1 |
| Protein Name | Mu-type opioid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 4,568
- Clinical molecules 14
- Avg pChEMBL 7.62
KEGG Pathways (5)
Active Molecules (4,568)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OKICQDFBWUMTDE
|
11.5 | Ki | 3 | — | |
RIAOSVMITNWHAH
|
11.4 | Ki | 3 | — | |
WPSMFHOVBQABMZ
|
11.0 | Ki | 3 | — | |
YCCQBABDNDRWSN
|
11.0 | Ki | 3 | — | |
RATBBTRECYJTEP
|
11.0 | Ki | 2 | — | |
ZHVLHUNBLJWDPM
|
10.9 | IC50 | 3 | — | |
FRPRNNRJTCONEC
|
10.9 | Ki | 3 | — | |
RIAOSVMITNWHAH
|
10.9 | Ki | 3 | — | |
WPSMFHOVBQABMZ
|
10.9 | Ki | 3 | — | |
RVZGUKSMLSUDCG
|
10.8 | Ki | 2 | — | |
RUMQBVLWLNKHTD
|
10.8 | Ki | 3 | — | |
KZEWGAHUIUQCHU
|
10.8 | Ki | 3 | — | |
NCZLAKYCTAUJMN
|
10.7 | Ki | 2 | — | |
MLQRZXNZHAOCHQ
|
10.7 | Ki | 3 | — | |
MOYUSPFIZGSIFO
|
10.7 | Ki | 3 | — | |
WTIFKSFIQUZRRN
|
10.7 | Ki | 2 | — | |
YDSDEBIZUNNPOB
|
10.6 | Ki | 4 | — | |
PPVICXFDCXSVFQ
|
10.6 | Ki | 3 | — | |
WYSHZXGBFZDQRH
|
10.6 | IC50 | 3 | — | |
UJSYTVDGBUQRBX
|
10.5 | IC50 | 3 | — | |
JPZJRCXPCGZJCY
|
10.5 | Ki | 2 | — | |
VMGFMOIZZDBILY
|
10.5 | Ki | 3 | — | |
QBPGLGPDPFXICV
|
10.4 | Ki | 3 | — | |
JQERUKPESNWSQA
|
10.4 | Ki | 2 | — | |
RDZUOGAZZXZDPY
|
10.3 | Ki | 3 | — | |
CBPOZLIYAVCTOE
|
10.3 | IC50 | 2 | — | |
DENICFHULARDRG
|
10.3 | Ki | 3 | — | |
IPPUMPUWHRNDMW
|
10.3 | Ki | 2 | — | |
RYIDHLJADOKWFM
|
10.3 | Ki | 3 | — | |
SEDKKDAEQSQWMA
|
10.2 | Ki | 2 | — | |
FRPRNNRJTCONEC
|
10.2 | Ki | 2 | — | |
KEYYWKJLTWUQSG
|
10.2 | Ki | 3 | — | |
LOCONFNPDMGOBD
|
10.2 | Ki | 3 | — | |
NLBUEDSBXVNAPB
|
10.2 | Ki | 3 | — | |
NLBUEDSBXVNAPB
|
10.2 | Ki | 3 | — | |
JPHBARUGZJTJNG
|
10.2 | Ki | 3 | — | |
NIZSYPMUUIDCPJ
|
10.2 | IC50 | 3 | — | |
KBYBCTDWHXSJNI
|
10.1 | Ki | 3 | — | |
FFBZQZXSTZLCDJ
|
10.1 | Ki | 2 | — | |
KOXWKZKLXNZQAO
|
10.1 | Ki | 3 | — | |
UVUFQEMGPJPSIS
|
10.1 | Ki | 3 | — | |
XREFQBQBSMEQOG
|
10.1 | Ki | 3 | — | |
XREFQBQBSMEQOG
|
10.1 | Ki | 3 | — | |
GARXJOUQUSNOGK
|
10.1 | Ki | 3 | — | |
GARXJOUQUSNOGK
|
10.1 | Ki | 3 | — | |
GWAMGWDJCYIREE
|
10.1 | Kd | 20 | — | |
IWBMAAUPHUCYCI
|
10.1 | Kd | 20 | — | |
LWMXWHIOMHIBJP
|
10.1 | Ki | 3 | — | |
MODBIBJHAWXYOZ
|
10.1 | Kd | 20 | — | |
ZRQMUCDHVVOENY
|
10.1 | Kd | 17 | — |