Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
FZTMDWIJTHPEMP 7.6 Ki 4
GSQPHXFZLYFUQD 7.6 Ki 2
IGXXJZSHANKJAD 7.6 Ki 2
JHJPBZPNRYMQKP 7.6 Ki 2
KLBQZWRITKRQQV 7.6 IC50 25 Yes
LSHDMKHXFDYKLP 7.6 Ki 2
QIUVHPATBGGVRR 7.6 Ki 2
QKRCVHKKBOUVNT 7.6 Ki 3
QQODNMGQNZBOAF 7.6 Ki 2
RIEFZSRXHBEIFW 7.6 Ki 2
VVGXLRREHSRFOF 7.6 Ki 3
XNPQDIOALLTRKK 7.6 Ki 3
YANGEESWIGIKOP 7.6 Ki 4 Yes
PVISFTMIHRDVDS 7.6 Ki 3
PVISFTMIHRDVDS 7.6 Ki 3
XCCCRVPCDJNFIY 7.6 IC50 2
ACTVOFFLDWZANE 7.6 Ki 3
CJGNMVAAMQAWEF 7.5 Ki 16
DMQAXIJUTYJHIV 7.5 Ki 6
GDLIGKIOYRNHDA 7.5 IC50 24 Yes
YVJCOHIKEMZVAO 7.5 Kd 4
IYRFHZMJBBCIFA 7.5 Ki 4
MBQMCWRJVSGZMF 7.5 Ki 2 Yes
NTBSVMCWAHSWAK 7.5 Ki 2
FJLHVGCNLNMUSS 7.5 IC50 5
VGIGHGMPMUCLIQ 7.5 Ki 12
AYPGYVOWMUSFPT 7.5 Ki 2
BEAHZBHBRZMAIL 7.5 Ki 4
DIXSEWSBXAEKKY 7.5 Ki 2
FSQHSKMGRAIYLO 7.5 Ki 3
GKKOWDZJMOVEBY 7.5 Ki 2
GPWMNUXSJDSCAV 7.5 Ki 4
KCLONPRRKHVPLU 7.5 Ki 2
MFJWXRIWIGLCGD 7.5 Ki 2
NQTXEWZDVUMZDO 7.5 Ki 2
PHHPFXWDLDXLPN 7.5 Ki 2
QVLZVRFIGXNZMN 7.5 Ki 2
VHHWNRROUCRXSK 7.5 Ki 3 Yes
WKNWCTUFTMDACE 7.5 Ki 2
ZJZRPZBCQDGSLP 7.5 Ki 3
PMXMIIMHBWHSKN 7.5 Ki 19
KUCRPWOVGMMXDP 7.5 Ki 3
LGHLMADLDHUIJY 7.5 Ki 7
QWGDMFLQWFTERH 7.5 IC50 23 Yes
RAPZEAPATHNIPO 7.5 Ki 28 Yes
MZCGNTZTYZJMJK 7.5 Ki 2
PSYAJOBNPBYKRW 7.5 Ki 5
DXJUCAUQIHNOAF 7.4 Ki 6
FDMSDOGSWFZXHI 7.4 Ki 2
HBMJSEBYZIMZIK 7.4 Ki 2
2D structure