Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
GEDGEGJCGBTAON 7.8 IC50 5 Yes
CIAWHNGOFJZBCL 7.8 Ki 5
ZZVUWRFHKOJYTH 7.8 Ki 11 Yes
LDPRUJUFFYEDJC 7.8 Ki 2 Yes
ITBDDOYXQTUJHV 7.7 Ki 4
KNZNKJDEMHGXSO 7.7 Ki 6
KNZNKJDEMHGXSO 7.7 Ki 6
FITQSJBSXMDHOS 7.7 Ki 4
FKKPXTRMLVLGJG 7.7 Ki 7 Yes
TVGLBSUFYKPBIU 7.7 Ki 2
WIKYUJGCLQQFNW 7.7 Ki 23 Yes
YKSKLZDPBLSMIO 7.7 Ki 2 Yes
MHNSOBBJZCWUGS 7.7 Ki 3
SWFSQSZMVIJILA 7.7 Ki 2
CLQMFOOMFPNKNA 7.7 Ki 3
CYAXTHULEFHIMG 7.7 Ki 2
DCPIUFZZSDRFTC 7.7 Ki 2
DFOFEBXXZMVAGG 7.7 Ki 2
GDRRHBZSXZXDLL 7.7 Ki 2
GJQONOYIKURBSD 7.7 Ki 3
HFWLILWGBZWYRI 7.7 Ki 2
KPWSJANDNDDRMB 7.7 Ki 17
LKFICSFQSQYFJF 7.7 Ki 2
MUPZZNZQFUCJBT 7.7 Ki 2
NWUBEEIEKUQVJL 7.7 Ki 2
PBFDUYRSNDQIDN 7.7 Ki 13
PPABRKQHBMJESP 7.7 Ki 2
PXQMPHKMJWQPRD 7.7 Ki 2
QLOCEFPHCAKSLE 7.7 Ki 4 Yes
RHTRBRRAADVASO 7.7 Ki 4
SKOALCKWENTDHG 7.7 Ki 3
UOWPMQNCLJZBEA 7.7 Ki 2
VDFDTTRCUDMUDX 7.7 Ki 2
YGYJEYXHZXOPGM 7.7 Ki 2
ZLPRNWIDJZJYMH 7.7 Ki 2
ZXFALDNPMLUADA 7.7 Ki 4
BCGWQEUPMDMJNV 7.7 Ki 30 Yes
LERNTVKEWCAPOY 7.7 Ki 6
PLDUPXSUYLZYBN 7.7 Ki 22
ZYRROKHYEJZYKQ 7.7 Ki 2
FHPIXVHJEIZKJW 7.7 Ki 18 Yes
WYSUFWVVSZJQRM 7.7 Ki 3
KPWSJANDNDDRMB 7.6 Ki 9
YFSPFZNLWSGJJK 7.6 Ki 6
AMEQLQYPRVOFMB 7.6 Ki 2
ATPAZLJUTRYFNR 7.6 Ki 2
CCJZAFYMSHLKFH 7.6 Ki 2
DERZBLKQOCDDDZ 7.6 IC50 20 Yes
DJGWTFPDOGEBKS 7.6 Ki 2
FCRIMCQUUZFBDN 7.6 Ki 2
2D structure