Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
ZFUMGFQOKSXSLS 7.9 Ki 2
ZTXJDBYCWAXXCA 7.9 IC50 3
XMXHEBAFVSFQEX 7.9 Ki 17
AMQPWRCXJRAWTN 7.9 Ki 2
IKBGPCPPFWCFRO 7.9 Ki 2
IZRPKIZLIFYYKR 7.9 Ki 3
JPDUMUHTXIBGHJ 7.9 Ki 3
JQNSYTMOXNMQTB 7.9 Ki 4
KOUMCBHTVFDPSI 7.9 Ki 2
NDXPOARUSJMOJN 7.9 Ki 2
RRMGPLJQTAJCCP 7.9 Ki 3
UZFUMFWJEGINFP 7.9 Ki 2
WVFQWSQTENHWCH 7.9 Ki 4
OOKYVXRSZPRVKD 7.9 Ki 2
QNFZIIFWVLXBEK 7.9 Ki 2
VEBMDYHKIXNRCE 7.9 Ki 2
WJRQBWWXQLYJAC 7.9 Ki 2
XRVALSGPOMRRRG 7.9 Ki 2
XVPCNLFLONEJBF 7.9 Ki 2
ZQADELCMZHYIPT 7.9 Ki 2
UOSUONQDJGNZCQ 7.9 IC50 3
UVKZSORBKUEBAZ 7.9 IC50 13 Yes
KUCRPWOVGMMXDP 7.8 Ki 3
RHPCETHLGGFAQB 7.8 Ki 9
TVKCCIBAUDHHBL 7.8 Ki 2
VAZUGKPZFFMBMS 7.8 Ki 2
WLCVFIFUKJWBRL 7.8 Ki 2 Yes
RTEBNFQOFLORPE 7.8 IC50 3
IRIGJBAWLKWASO 7.8 IC50 3
XRYLGRGAWQSVQW 7.8 Ki 4
BXUKKRHEMKVWOY 7.8 Ki 4 Yes
CCXXDPNVVABEGJ 7.8 Ki 2
CGPUMTTUBWGRHT 7.8 Ki 2
FAXDKDSDNWXAIS 7.8 Ki 3
FIMFEAXKPOZWDG 7.8 Ki 4
HKPKDTNLXGOYIC 7.8 Ki 4
IGYNNXYCDMNULT 7.8 Ki 2
LDUDMYAXGOQOGO 7.8 IC50 3
MNSGCVNHLLGCDG 7.8 Ki 2
MNZXCYDDVWTITD 7.8 Ki 3
PCRWWFINVOSHRN 7.8 Ki 2
QAXGZLPJWOSHHV 7.8 Ki 2
REXVRCXDIWIKGL 7.8 Ki 4 Yes
STXMJDYUJFBELE 7.8 Ki 2
VDNHGXHYXNDCOW 7.8 Ki 2
VNYAKKUPVDUAEG 7.8 Ki 2
WCXUWQZNCRRRDD 7.8 Ki 2
WRWUGHDNJYUGGD 7.8 Ki 3
KLBQZWRITKRQQV 7.8 Ki 21
VPZDYZMLWKUTOB 7.8 IC50 2
2D structure