Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
QJPBTFRGWJLPSI 8.2 Ki 2
YRDKYTTYDOWYLC 8.1 Ki 5
ZPEIMTDSQAKGNT 8.1 Ki 35 Yes
DXJUCAUQIHNOAF 8.1 Ki 2
LGHLMADLDHUIJY 8.1 Ki 7
OHBPVXVMMZZMKM 8.1 Ki 2 Yes
FSRSEANZUZHDHK 8.1 Ki 2
DREBLEJJYUKNLT 8.1 Ki 2
DWIXBLOYUJIYNT 8.1 Ki 6
KVHHUZUNLIGTBY 8.1 Ki 10
RGCVKNLCSQQDEP 8.1 Ki 16
RGQXJYRGDMABLT 8.1 Ki 3
RUWZQSJWDUNAEU 8.1 IC50 3
UEMKNKCKJCNUSX 8.1 Ki 2
ZFVQRQOPWCBDOI 8.1 Ki 2
BQDBKDMTIJBJLA 8.1 Ki 5
ZCRCTVHOBQJBNB 8.1 Ki 2
OZVCVTCZRYMODR 8.1 Ki 3
LWOMEPYLSGEMDX 8.1 Ki 2 Yes
ZKIAIYBUSXZPLP 8.1 Ki 29
KJQCJXUDPPZASI 8.0 Ki 2
RUKTXHCGSFMYLO 8.0 Ki 3
AITHPZKEMCVCDZ 8.0 Ki 2 Yes
CEXVQARQHVKRBU 8.0 Ki 3
MJJALKDDGIKVBE 8.0 IC50 30 Yes
ZUSSMNOENOGGGY 8.0 Ki 2 Yes
CPNTXNSOEZESIH 8.0 Ki 4
CPNTXNSOEZESIH 8.0 Ki 4
DLONTNINHYMHFB 8.0 Ki 2
IJMPFBJUROFOGZ 8.0 Ki 4
IJMPFBJUROFOGZ 8.0 Ki 3
JTCQOAITNDJYSA 8.0 Ki 3
JTCQOAITNDJYSA 8.0 Ki 3
NWCYKTKORNLIRC 8.0 Ki 3
ODKRBJGIPOQDPJ 8.0 Ki 2
ROQGCKBWSKAVEH 8.0 Ki 2
SAKVKDBLCRHLAV 8.0 Ki 4 Yes
SECXHJRGBAZUCO 8.0 Ki 4
XSZZVXRYXJUWCA 8.0 Ki 3
XSZZVXRYXJUWCA 8.0 Ki 3
YANGEESWIGIKOP 8.0 Ki 7 Yes
ZHYJMAJSBAQRIU 8.0 Ki 4
ZHYJMAJSBAQRIU 8.0 Ki 4
AWYSEPZPTVMKBT 8.0 Ki 4
LCKBEOTXTNWYRG 8.0 IC50 8 Yes
URKOMYMAXPYINW 8.0 Ki 27 Yes
CZXWYWSRENNIBD 7.9 Ki 2
JUQLTPCYUFPYKE 7.9 Ki 25
QOYHHIBFXOOADH 7.9 Ki 16
XRYLGRGAWQSVQW 7.9 Ki 3
2D structure