Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
LMBAXHGIFALPQJ 8.3 Kd 4
MODBIBJHAWXYOZ 8.3 Kd 20
MWNWERUECAJGJC 8.3 Kd 6
NNBLASKQLZCYBL 8.3 Kd 4
OJYUKAHOHYUAHF 8.3 Kd 6
ONVSJLPIADFJKR 8.3 Kd 4
OVYZCEIGUJNWKN 8.3 Kd 4
PCFGLLVVPCPPIG 8.3 Kd 4
PKALTNFRHBJDRH 8.3 Kd 6
QVAKGXNPTKFJST 8.3 Kd 6
RHRPOJKRNUHOJA 8.3 Kd 4
RXDHWPCPLSUTCP 8.3 Kd 4
SAEILUJHGHNPAN 8.3 Kd 4
SRELLSOOXBJTLE 8.3 Kd 4
UAFKZBOQJUSIDU 8.3 Kd 4
USBWQDPYNKDRSV 8.3 Kd 4
UWTPDHDYCBTOMN 8.3 Kd 4
XNSQSOGNTZGMDA 8.3 Kd 4
XQOLXGFKFIWXQP 8.3 Kd 6
YPAOZTCVMTXDID 8.3 Kd 4
YYXYUTGQFNFTGX 8.3 Kd 4
ZKKBZRDZTBXDKE 8.3 Kd 4
ZYFQYFZOSKEOGJ 8.3 Kd 4
VILNAIPEYFWQQH 8.3 Ki 2
DTYDZUZTWZDAGL 8.3 Ki 3
FLTAIVXWWOKLBO 8.3 Ki 2
QNNXKPSMUIHGIZ 8.3 Ki 2 Yes
SUHCNXHLKUQVER 8.3 Ki 2
URSKGEZFWCRYMD 8.3 Ki 3 Yes
VLUYCVQWTQUWPI 8.3 Ki 2
VTIFNIOOCLEWLJ 8.3 Ki 2
XJGVXQDUIWGIRW 8.3 Ki 17
HNJJXZKZRAWDPF 8.3 IC50 7
IEMJYQZKJFERDW 8.2 IC50 5 Yes
LDAIZSJPULESPS 8.2 Ki 2 Yes
FPDIERBPQFAFSI 8.2 Ki 17 Yes
KTWZXHKXAGXWOB 8.2 IC50 3
LGIIUKGHECNJNZ 8.2 Ki 2
WSAMXDVPPULVBH 8.2 Ki 3
ZDIGNSYAACHWNL 8.2 Ki 2
CXDSZAINFKAKPN 8.2 Ki 4
OIZYYUJMNZAXNN 8.2 Ki 3 Yes
RMQXJQUUIKBXMM 8.2 Ki 2
UMSPPMMERAOIRT 8.2 Ki 2
XBJQRDCFABQBGT 8.2 Ki 3
FBCSWIXKXHSYBN 8.2 Ki 18
BTSCZNWXJQSJIE 8.2 IC50 10
BTSCZNWXJQSJIE 8.2 IC50 10 Yes
YGQQBKYVKLZEMA 8.2 Ki 2
IMKMPTLRTHMERW 8.2 Kd 4 Yes
2D structure