Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
SHNQYDFOONPSKV 8.5 IC50 3
URZPDWAADSKBHJ 8.5 Ki 3
WZMVQZJKOVPVGZ 8.5 IC50 4
KVWDHTXUZHCGIO 8.5 Ki 32 Yes
AWKFJGDSZGEFRY 8.5 Kd 4 Yes
YVENIGOVHPMTDH 8.5 Ki 23
ZOYPHDPQFYRSLG 8.5 Ki 2
LFSBNTMFCXGIEC 8.5 Ki 2
JHZAKXOZEGDRAJ 8.5 Ki 4
OSJJYEUEJRVVOD 8.5 IC50 17 Yes
VTMJTHCQLMVWGT 8.5 Ki 4
GKDBTHSYQZTDAJ 8.5 IC50 13
RUKTXHCGSFMYLO 8.5 Ki 3
QBUBIPIOMZYFEI 8.4 Ki 2
ACTVOFFLDWZANE 8.4 Ki 3
YZIDTWIJPIHTCE 8.4 Ki 3
PWJDUASUWRTROR 8.4 IC50 3
CVUXESFCUHCXHB 8.4 Ki 2
IQWBKNWLBVZZLG 8.4 Ki 2
BYPMJBXPNZMNQD 8.4 Ki 18
GQWSXILTLUTBAJ 8.4 Kd 4 Yes
IYDOAHOHMRQFTJ 8.4 Ki 4
MAWNODXTLNGOAA 8.4 Ki 2
NANQRVOKMXDMNL 8.4 Ki 2
SKXJKSJHHFLVAP 8.4 Ki 2
WBCSOAILRDZMDJ 8.4 Ki 2
YSQQOGOBORIIMG 8.4 Ki 2
ZWZGWXZGAUJLHN 8.4 Ki 3
OWMBYQVIMDTSAW 8.4 Ki 2
ZMOPTLXEYOVARP 8.4 Ki 14 Yes
KWUQZAPLAOREKL 8.4 Ki 3
RHPCETHLGGFAQB 8.4 Ki 9
LSOVNGNFKVHURS 8.4 IC50 2
BIJXMFDKONGOAN 8.3 Kd 4
BQYXPJXIOSEURA 8.3 Kd 4
CDGJSIMJNZNZFE 8.3 Kd 6
CDZGYTJJJXXWBS 8.3 Kd 4
DDBBPVWZBRHZDD 8.3 Kd 4
FARKBYHYALPKMO 8.3 Kd 4
FASDKYOPVNHBLU 8.3 Kd 9
GHZHZIJXYOTTAA 8.3 Ki 2
GWAMGWDJCYIREE 8.3 Kd 20
HKCHNLZUCRQSTO 8.3 Kd 4
IOSVPGDHSQVBED 8.3 Kd 6
IWBMAAUPHUCYCI 8.3 Kd 20
KCCBFGKNVMTXIQ 8.3 Kd 6
KGGHECZDYBMALC 8.3 Kd 6
KIRWEWNKOWMEBM 8.3 Kd 4
LDXAOQSIBXRCIN 8.3 Kd 6
LKPZDFCAQDGUKZ 8.3 Kd 4
2D structure