Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
NRNPLYWFPSCQAF 8.8 Ki 3
RONZAEMNMFQXRA 8.8 Ki 9 Yes
YEFYNZHDZSJWCN 8.8 Ki 3 Yes
ZAIFESHMEUUZQE 8.8 Ki 3 Yes
ZUXABONWMNSFBN 8.8 Ki 29
QSLMDECMDJKHMQ 8.8 Ki 20
KYIGOCCCBXRHNJ 8.8 IC50 43
UEQUQVLFIPOEMF 8.8 IC50 21 Yes
YVEWHDHDFNFTCD 8.8 Ki 2
QBPDZEVGAGDUQY 8.8 IC50 3
SFOPQOZLZFKLOD 8.8 Ki 4
DDHSIUUOIYFUOU 8.7 Ki 2
SLVMESMUVMCQIY 8.7 Ki 14
PTZUOUKVZMOWMQ 8.7 Ki 3
YECBIJXISLIIDS 8.7 Ki 7
QZUDBNBUXVUHMW 8.7 Ki 39 Yes
FPCCSQOGAWCVBH 8.7 Ki 16
IVQAEXPSYGMKTP 8.7 Kd 2
JWDZDXFXHWMSGR 8.7 Ki 3 Yes
YDNXGTGGTKAMFI 8.7 Kd 2
ZQDWXGKKHFNSQK 8.7 Ki 3
DXJUCAUQIHNOAF 8.7 Ki 5
GXDALQBWZGODGZ 8.7 Ki 21 Yes
RJAXVZUSTIFVGP 8.7 Ki 2
YRRXDGSRIMGDFU 8.7 Kd 2
SOYKEARSMXGVTM 8.7 IC50 8
FLZIWHXEHDCVMN 8.7 Ki 2
PKONXOYDGGORHO 8.7 Ki 2
QKNADAQNYDFJFJ 8.7 Ki 2
UJLZUVUUHZVHFF 8.7 Kd 2
JTLCTTWVUAIQHD 8.6 IC50 17 Yes
LHTXSHOSMCEFFX 8.6 IC50 3
SWFSQSZMVIJILA 8.6 Ki 3
GIEBQTVDYXTBCS 8.6 Ki 2
GPVDPKZTACUYNW 8.6 Ki 3
LDMXQNXCFMLIER 8.6 Ki 2
VKVAJQSZVWNRMB 8.6 Ki 3
GWVFJNPANMKQSY 8.6 Ki 2
LPHIWCBAJGQIIF 8.6 Ki 3
NZFSPDVTABQASR 8.6 Ki 3
OEYDBWKMXFZENQ 8.6 Ki 3 Yes
SUYKBMCECCINPJ 8.6 Ki 2
KNZNKJDEMHGXSO 8.6 Ki 6
MSQRTETUBFIHMP 8.6 IC50 9 Yes
GETROLYXSDDSDH 8.6 Ki 2
PVLJETXTTWAYEW 8.6 Ki 2
AAGWAYIWKWJZAD 8.6 Kd 3
PCLYKAGGELJIIV 8.6 Ki 4
SULKMHQPINMVTR 8.5 Ki 2
HMWYNGSUVFCIHB 8.5 Ki 2
2D structure