Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
RZBPSXCZVILRNE 9.2 Ki 4
ABDWUBPDHWDFCV 9.2 Ki 2
ACTVOFFLDWZANE 9.2 Ki 3
VVYQHHROMNFSAO 9.2 Kd 4
LXGZSTDLYCGLAE 9.1 Kd 4
IAFSRSYSLPAOJE 9.1 Kd 2
HPVUAGMZZRSSHI 9.1 Ki 2
LDKQFEPUPKIHCG 9.1 Ki 2
YMFHXRKTKHBRIX 9.1 Ki 4 Yes
RPUXCIYWJSVFFV 9.1 Ki 6
ITEQLSGAAAJLOU 9.1 Kd 2
AXIFLPLKZRNVDP 9.1 Ki 2
HILDNLJIJXAVHA 9.1 Ki 3
NZEFYLGMSWSUDH 9.1 Kd 4
YZAHEHXQIMZHAJ 9.0 Ki 5
BFEIADQANSGVFP 9.0 Kd 2
FRUMSZUUBXPHHF 9.0 Ki 4 Yes
NZGLSOKQCCNTMG 9.0 Kd 2
PYSIAKZWZJNMNM 9.0 IC50 2
VSWBSWWIRNCQIJ 9.0 Ki 2
VSWBSWWIRNCQIJ 9.0 Ki 23
YFGUGMIFVSSOJY 9.0 Kd 2
YKMYFJKVCCQVAY 9.0 Ki 2
YLWRKTVVIPNRDE 9.0 Ki 4
ZCVMWBYGMWKGHF 9.0 IC50 19 Yes
GIJXKZJWITVLHI 9.0 IC50 16
GQDIAXARFJUVLN 9.0 Ki 4
JJKMOFKIYHXREY 8.9 Kd 5
PTVITZRFRXZZEA 8.9 Kd 4
MBUVEWMHONZEQD 8.9 Ki 17 Yes
WWZJPGCAXYFHPB 8.9 Ki 4
BSOLCASXROXPRZ 8.9 Ki 9
DYRUSALPYKCZDY 8.9 Ki 3
VIEHHRQCEMIKCL 8.9 Ki 2
JJCFRYNCJDLXIK 8.9 IC50 25 Yes
VLAMSHNLMPNZGJ 8.9 Kd 2
DGZLHXBKGBELTQ 8.9 Ki 4
PSVLBKXIZLIMQR 8.9 IC50 3
ZQXPNWSXFWKXRZ 8.9 Ki 2
JAUOIFJMECXRGI 8.9 IC50 13
WYSUFWVVSZJQRM 8.9 Ki 4
BSOLCASXROXPRZ 8.8 Ki 9
GMIVYDCUSUDJGH 8.8 Kd 2
HDOZVRUNCMBHFH 8.8 Ki 26 Yes
IYRFHZMJBBCIFA 8.8 Ki 4
UHPLDFSEISHDBD 8.8 Ki 2
UUEDQZRCAVWNIH 8.8 Ki 2
ZSCDBOWYZJWBIY 8.8 Ki 2
AVFYUSOOXDDQAW 8.8 Ki 2
MCVGJQYUOLRXOM 8.8 Ki 3
2D structure