Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
AUTKMGMMFJXIDV 6.8 Ki 2
QTDHTTNBIMOVCI 6.8 IC50 5
FPVHORFNDSKMPV 6.8 IC50 5
JPXQQLVVAAHNSC 6.8 Ki 7
YQNWZWMKLDQSAC 6.7 Ki 15
ZBUWQTCXTJMDCD 6.7 Ki 2 Yes
SJEXSMOVRPPLBZ 6.7 Ki 8
SJEXSMOVRPPLBZ 6.7 Ki 4
CILDROBPHGWMGB 6.7 Ki 6
JCCNYMKQOSZNPW 6.7 Ki 4
MVKKLGNVARQKRP 6.7 Ki 13
ZFUOLNAKPBFDIJ 6.7 Ki 7
ZFUOLNAKPBFDIJ 6.7 Ki 7
ZZEQOXMRTJPRMI 6.7 Ki 2
AIYDXOYEOAYSGJ 6.7 Ki 4
GEICAQNIOJFRQN 6.7 Ki 3
KVJXXDNXTCGJKY 6.7 IC50 5
FPAJMJGGDZGJPZ 6.7 Ki 2
GIZCWMURBFLMON 6.7 Ki 4
GSUXFSXZSCBDQK 6.7 Ki 2
JMGBVGDZPLNFAE 6.7 Ki 2
NFCYQBPNSWBYEF 6.7 Ki 4
NXHYSNCNFYHMIU 6.7 Ki 2
TYDWSEQLTIBAPO 6.7 Ki 2
UZJWAFOJOSGEKL 6.7 IC50 15
YRZFLXOYFQEHFH 6.7 IC50 3
IYRFHZMJBBCIFA 6.7 Ki 4
UCQNMJXTWOYVNH 6.7 Ki 6
ANTSCNMPPGJYLG 6.7 Ki 7
SQGWMVXOYSHVTI 6.7 Ki 6
ZIWFCOIGUNPHPM 6.7 Ki 5
IESJRUUOIHDONG 6.7 Ki 8
HBRHULDGKNIFGB 6.7 Ki 4
QNKGTIWNFNPEJL 6.7 Ki 11
DMULVCHRPCFFGV 6.6 IC50 10
WWZJPGCAXYFHPB 6.6 Ki 4
JNUCCWMHZZUFKE 6.6 Ki 2
BTSMIVQFEUCDAW 6.6 Ki 8
ADUYXHYSTCIMEO 6.6 Ki 7
JOZMHQIYXRYITJ 6.6 Ki 2
MBMAQWYADJFPMU 6.6 Ki 2
MCWADYMQWQHSRA 6.6 IC50 5
MHAQTEBGBYFXKL 6.6 Ki 2
VGLVSBTUAYHUEF 6.6 Ki 2
ZENBFJWQHFZSBC 6.6 Ki 2
BETHXCLHMRGYBW 6.6 Ki 9 Yes
BPDDCCYSOYRMEC 6.6 Ki 8
JVCJWEYSNNCGKX 6.6 Ki 3
DARWEDNPGILOPQ 6.6 Ki 2
IFPGADOWNOXLNQ 6.6 Ki 6
2D structure