Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
FGTGRXMIFIZGBG 6.9 Ki 10
IMEKNFSOCZJKQI 6.9 Ki 4
VTMJTHCQLMVWGT 6.9 Ki 4
SFOPQOZLZFKLOD 6.9 Ki 4
PHLBKPHSAVXXEF 6.9 IC50 12
VKNIGNGTZIYLFI 6.9 IC50 5
BOOQTIHIKDDPRW 6.9 Ki 14
CSSKAGWIWQOQME 6.9 Ki 2
IIRIKFXWBJTDCC 6.9 Ki 3
IQNSUCJNGFOYPQ 6.9 Ki 2
LQEATNFJCMVKAC 6.9 Ki 14
MANRLQSCJCTMOZ 6.9 Ki 2
MNHDKMDLOJSCGN 6.9 Ki 23
PREVLKLSVWYCAY 6.9 Ki 2
REJVZJBLJWRHQL 6.9 Ki 2
RTMHXVRCXRAHLV 6.9 Ki 3
RUMOWLXMMCFECC 6.9 Ki 2
VRBKIVRKKCLPHA 6.9 Ki 22
WWZJPGCAXYFHPB 6.9 Ki 4
XMFRRROSDAWYLB 6.9 IC50 5
XNVKJWRHFRDBHD 6.9 Ki 4
XPRWZTNAGMLCGT 6.9 Ki 2
GZKLJWGUPQBVJQ 6.9 Ki 24 Yes
OOGJQPCLVADCPB 6.9 Ki 9
QLTASWSCCMMISJ 6.9 Ki 4
ZTBBOIYRZHAFIN 6.9 Ki 8
UOXWVJAPLQMAAN 6.9 IC50 5
YVUQSNJEYSNKRX 6.9 Ki 36
SNZBWZJDHITSSV 6.9 Ki 3
OWPHKTVZEZNCMB 6.9 Ki 2
PWQSSAWBTAKELO 6.8 Ki 2
QVYRGXJJSLMXQH 6.8 Ki 14
FAIMGWSOSCFGRU 6.8 IC50 6 Yes
GKTQBPYMIGXPKG 6.8 Ki 21 Yes
GKTQBPYMIGXPKG 6.8 Ki 18
GLXQEUGDWMYWCC 6.8 Ki 2 Yes
HXBMOXWVYIRYHK 6.8 IC50 2
FGXWKSZFVQUSTL 6.8 Ki 10 Yes
AQVKRBFXFFKXJV 6.8 Ki 2
CWXOTCCLEKNUJY 6.8 Ki 2
DBFNYFZBHMQFLI 6.8 Ki 2
JQEQULOLEPTBRS 6.8 Ki 3
KWZBJWOQFABHPF 6.8 Ki 10
NMLHPAJBQUFHAV 6.8 Ki 2
NTYJJOPFIAHURM 6.8 IC50 4
RFDSGHNJJQPTLS 6.8 Ki 2
ROKAKGMAWJNFEN 6.8 Ki 6
CFGLHQSIGAVKRU 6.8 IC50 5
NSMCYUMPIGJKHV 6.8 Ki 9
NDWXGJDJKXDMOV 6.8 IC50 3
2D structure