Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
UCNOTTVNPRSTFW 7.1 Ki 8 Yes
HQUSWISCKAODEN 7.1 Ki 5
LDAHGSIPSNYPMF 7.1 IC50 5
ALTKABGEMCJWJH 7.1 Ki 15
BBQVIKFUQPNVLK 7.1 Ki 4
FEIOPVQTLJUJBR 7.1 Ki 2
IGZMIXBCHNOMPG 7.1 Ki 2
LLEJNWFSXZIFMW 7.1 Ki 2
MOHMWXTYADLKCG 7.1 Ki 2
PDJBLXDNFLXACI 7.1 Ki 2
QLGIWKYNMSCERQ 7.1 Ki 2
RHDOFWFMSRHNFN 7.1 Ki 2
UFCXUUIZIMGORH 7.1 Ki 2
XHHDACAEDLRJOJ 7.1 Ki 5
YDHQRFQQOKRWAD 7.1 Ki 2
KHPOIBBWMVNTMI 7.1 Ki 5
OZVCVTCZRYMODR 7.1 Ki 4
SWGWJQBPCJEQJC 7.1 IC50 4 Yes
HCYAFALTSJYZDH 7.1 Ki 14 Yes
LJVNYCDXBXGQIK 7.1 Ki 14 Yes
NMALCZJKSYZTRE 7.1 Ki 7
SPMHWCSUNSWHDK 7.0 IC50 5
SVJMLYUFVDMUHP 7.0 Ki 26
KAXNWVHHUKHNDK 7.0 Ki 3 Yes
CDQRIIUMNLMHRH 7.0 Ki 6
VCADIWSEVTZZOR 7.0 Ki 3
AEWQIKDEAWAPPV 7.0 Ki 2
AJUWTQZJBKWQNV 7.0 Ki 2
AYWYOYAKLYFQAR 7.0 Ki 3
DADRXTGBZRBZMD 7.0 Ki 2
DCPIUFZZSDRFTC 7.0 Ki 2
FLTBEMVEAFMWDD 7.0 IC50 2
HLXZPGHNFUSVMT 7.0 Ki 2
JHJPBZPNRYMQKP 7.0 Ki 2
JWPAYBAIIARWMG 7.0 Ki 19
NHOMRPYETSURDH 7.0 Ki 2
OZCVIUHHOUTJJN 7.0 IC50 2
OZZLMZAQJKSGCB 7.0 Ki 3
SDPQHMHFTWVGGO 7.0 Ki 2
XRJGWSMTLAFHBN 7.0 Ki 21
YDRCHQQFHSPVMO 7.0 Ki 2
ZNOFXQRZLXBDTB 7.0 Ki 2
VMLLHZVDHFWOOM 7.0 IC50 3
OLJSGKYQYTWQNJ 7.0 Ki 2
XQDRWCFJBHLWPR 7.0 IC50 8 Yes
RLMGUPUESXPDFJ 7.0 Ki 5 Yes
OURPZJJZFFKVJH 7.0 Ki 10
QXYZJXCNTMMWEO 7.0 Ki 15
RKEGNNLTPLWIIC 7.0 Ki 2 Yes
JWYUBODPEUBFLH 7.0 Ki 11
2D structure