Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
IYAJUPFWKMPDJJ 7.3 Ki 4
JAWGTZDKZCZPKP 7.3 Ki 4
JHJPBZPNRYMQKP 7.3 Ki 2
JHZAKXOZEGDRAJ 7.3 Ki 4
JVDFBAQLTSMMBQ 7.3 Ki 2
LEHDCEDFGAFVGX 7.3 Ki 2
LQCZDIMQFUOGJG 7.3 Ki 2
NYWUAMYWDNANQG 7.3 Ki 3
OSUVEVWOPQLILG 7.3 Ki 2
QYAXGGUCDQSHIT 7.3 Ki 4 Yes
SHRVEEBUQYOBLS 7.3 Ki 2
UJDYUOWUTALBPP 7.3 Ki 2
VXQLVBTWUUQZBI 7.3 Ki 2
YDRCHQQFHSPVMO 7.3 Ki 2
YEGSREZTMOWGTG 7.3 Ki 2
YFTFPJHCROIDGR 7.3 Ki 2
YSGLQQUCJIOYSX 7.3 Ki 4
ZBUWQTCXTJMDCD 7.3 Ki 2 Yes
CHGXPKZHRZIZSQ 7.3 Ki 7
SMANXXCATUTDDT 7.3 IC50 25 Yes
DTYAFBJXWWLRMA 7.3 Ki 4 Yes
TZFKQPVOFBQHAZ 7.3 Ki 9
BKRGVLQUQGGVSM 7.3 IC50 26 Yes
CEUORZQYGODEFX 7.3 Ki 31
RQTZTSPFFYDZKA 7.2 Ki 5 Yes
NAGKIWFBALBSMD 7.2 Ki 2
CQGTWGRGLDAJSE 7.2 IC50 3
UNTNFKPMHAXOEK 7.2 Ki 7
CUIDNQSCWXAPRS 7.2 Ki 2
DMQWGZFKPDYZCH 7.2 Ki 2
DWNROPYUHGRJJG 7.2 Ki 2
FLDDBSYUKQDTDX 7.2 Ki 2
GJJRSPSNZFRQIQ 7.2 Ki 2
GPRHHSZIXIDKDN 7.2 Ki 3
GUOQPFNLBAXWIZ 7.2 Ki 7
HNLNXYUSMGCHFW 7.2 Ki 4 Yes
MYZGZNJBQOQRTJ 7.2 Ki 2
RMSWKUOSOVPFPF 7.2 Ki 2
VOPUEJLKUSXAOZ 7.2 Ki 2
WGNYIJNJSDBPLE 7.2 Ki 3
WLHRCQLHMHKOKG 7.2 Ki 2 Yes
YMYZSITWBGWUAF 7.2 Ki 2
ZEWQUBUPAILYHI 7.2 Ki 21
KEEXCUUQRQNRNF 7.2 Ki 3
PBYSLXLVOFLVAY 7.2 Ki 3
HXTGXYRHXAGCFP 7.2 Ki 6
KAHXPONUPROIRS 7.2 Ki 7
XHIUHIDIRNZTAW 7.2 Ki 7
GXZWKZAOGQRNTL 7.2 Ki 12
MVMQESMQSYOVGV 7.2 Ki 6
2D structure