Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
JASKXIBVQDMBJJ 7.4 Kd 4
MJDSQILVNHZQRV 7.4 Ki 2
MMEQHMVQEKIHIG 7.4 IC50 3
NDAMBUDREMDLPA 7.4 Ki 2
WFGYPTMXXGANAS 7.4 Ki 2
IMEKNFSOCZJKQI 7.4 Ki 4
VFCNPRIWDSWJIG 7.4 Ki 2
AQIZHUDMGJRAMJ 7.4 Ki 2
AQQFXOLTZFTABW 7.4 Ki 6
ASARBMLXIRIMCK 7.4 Ki 2
BACLISNXCXJOMR 7.4 IC50 4
GUGOEEXESWIERI 7.4 IC50 18 Yes
IBTMKWBYOYIWBF 7.4 Ki 2
LGNOCEJCJLXMEA 7.4 Ki 2
PXJLHYOGLFJGQN 7.4 Ki 2
QQERDUJEEYWVED 7.4 Ki 3 Yes
RRTCFJGKAMKAIY 7.4 Ki 14
RUCWOVBWUVMXEY 7.4 Ki 2
SEIOTCVWLCUESB 7.4 Ki 2
SOXIOTAVNTWQJT 7.4 Ki 4
TVBIHDSWRDFHAA 7.4 Ki 4
UUYDLXMNWLLYQV 7.4 Ki 4 Yes
VCLTUEPMXZBALZ 7.4 Ki 3
VFKIKYZNUCGJGD 7.4 Ki 3
VMTWXOTZXVFSPH 7.4 Ki 4
ZQVGMOFPWWNMNB 7.4 Ki 2
MSMKOTVNTGCTFQ 7.4 Ki 2
PCLYKAGGELJIIV 7.4 Ki 4
DMYWKEKMOKMLKU 7.4 Ki 2
FXHLGRYCQSRFHY 7.4 Ki 9
MKLCNRHAJGACTJ 7.4 Ki 2
MVWVFYHBGMAFLY 7.3 Ki 31 Yes
USGLWFZAXHASGB 7.3 Ki 4
DZXZPVGWRZCXDH 7.3 Ki 20
ODJIGTDOQQQJKM 7.3 Ki 3
OIXSYJAHIPQFMO 7.3 Ki 2
SXJNGGGCIYFZDT 7.3 Ki 2
HGLGWLWXYRAXPK 7.3 Ki 3
HPJNWYRQLUNOIA 7.3 Kd 4
PVWQFOKNAQZORV 7.3 Ki 2
ZNWOCPPAOLYORT 7.3 IC50 3
GQDIAXARFJUVLN 7.3 Ki 4
DVSMVUMYJDOPJQ 7.3 Ki 16
FGWSLMPEBIIYTF 7.3 Ki 2
GUUFVYCRQBZPLO 7.3 Ki 2 Yes
HDDLHPPRMNRBQB 7.3 Ki 4
IFFNPVFKAKKFAP 7.3 Ki 2
IGLADUDHPDHSRD 7.3 Ki 2
IRGGYSVFJCBILG 7.3 Ki 4
IUIGATKKQCOBAF 7.3 Ki 2
2D structure