Target Details
UniProt ACP35367
Gene SymbolHRH1
Protein NameHistamine H1 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 872
  • Clinical molecules 125
  • Avg pChEMBL 7.54
Top Co-occurrence Targets
Active Molecules (872)
InChIKey pChEMBL Type Targets Clinical
AYFAGRAOJPSHSH 10.2 Ki 19
MBVVVQZOMZFVJF 10.0 Ki 4 Yes
YNNUSGIPVFPVBX 9.8 IC50 24 Yes
UJMUXUJLIHKBEA 9.8 Ki 4 Yes
WYRUGBCTQBZIHO 9.8 Ki 5 Yes
ODQWQRRAPPTVAG 9.8 Ki 2
XRYLGRGAWQSVQW 9.7 Ki 7
HTHMMDLGLVQHEM 9.7 Ki 3 Yes
QTQRWXSELPXXAV 9.7 Kd 2
ODQWQRRAPPTVAG 9.7 Ki 20 Yes
GFOPLENUCATIPC 9.6 Ki 3 Yes
ODQWQRRAPPTVAG 9.6 Ki 14
REXDQAIKTDDWAC 9.6 Ki 4
WRGOSJVRKURGMQ 9.6 Ki 3 Yes
HSINSDXPTLWBKS 9.6 Kd 2
IBILQKIYEWGQDQ 9.5 Ki 2
DCGYGKIBQOAKTB 9.5 Ki 3 Yes
IKNJHFAJDYZLNM 9.5 Ki 2
OUEZWZJJIKBFFV 9.5 Ki 5
WYRUGBCTQBZIHO 9.5 Ki 3 Yes
HRSYZRFBUGIVHN 9.5 Ki 4
KCCUYRWFHHFONN 9.5 Kd 2
SXNOWQCFHNZUIX 9.4 Ki 4
UEQUQVLFIPOEMF 9.4 Ki 13
KGNWCYQCPGINGS 9.4 Kd 4
RPPOAMDDJXHPIC 9.4 Kd 2
VFIDGXZRONKQBZ 9.4 Ki 5
WCNMMPUKVKKLKP 9.4 Kd 2
MVMQESMQSYOVGV 9.4 Ki 3
ACTVOFFLDWZANE 9.4 Ki 9
CEJBRQBGHDEPNJ 9.3 Kd 4
CJMVJEMHSLDPMO 9.3 Ki 4 Yes
IMEKNFSOCZJKQI 9.3 Ki 5
LRTHKJMSTYBFFO 9.3 Ki 2
KMFDXNUGIFDFHQ 9.3 Ki 5
BSOLCASXROXPRZ 9.3 Ki 9
ACTVOFFLDWZANE 9.3 Ki 9
SAMYTBZVLLYSKN 9.3 Ki 5
YIJMYSUOYUNZGL 9.3 Kd 4
AMOACTSTZUXXDX 9.2 Kd 4
FRXWLMMHSBOBJK 9.2 Ki 3
ACTVOFFLDWZANE 9.2 Ki 3
BTFVTAWVFBWGHC 9.2 Kd 4
FNEORDYLRZOEEP 9.2 Ki 5
NSRMKMSTPLJNHM 9.2 Ki 6 Yes
OZUYIQYXHKJSCF 9.2 Kd 4
ULSSDVVGTBLGMG 9.2 Kd 2
UXQVMDVKHFQOEU 9.2 Ki 5
WXPNDRBBWZMPQG 9.2 Ki 28
MVMQESMQSYOVGV 9.2 Ki 6
2D structure