Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
PNMMHGYXIWNCEE 8.8 Ki 4
QUGYQBYWGZYWAK 8.8 Ki 3
RFEHYTXXQXNSOO 8.8 Ki 3
YCKRBYBOMGAOET 8.8 Ki 2
ZEGBQBDRCBJTSW 8.8 Ki 2
BGFYEOBLDYCILL 8.8 Ki 4
KAHFZGUOPFFVHW 8.8 Ki 4
KTSCUAMGSPLOJT 8.8 Ki 3
KYBQSIXBWBXIFN 8.8 Ki 3
MDOKTLACQIDXQG 8.8 Ki 4
MRCKSWXOWOMYII 8.8 Ki 3
NTYDVUXIVLYUEG 8.8 Ki 3
OQDVCLJHYBLHNT 8.8 Ki 2
QPOJVLKZPPBFKN 8.8 Ki 3
RONZAEMNMFQXRA 8.8 pIC50 9 Yes
SOUVKJLYRGDDOT 8.8 Ki 3
UDYXSPVICNNUPJ 8.8 Ki 9
NHANMZHYPOUORL 8.8 Ki 4
XTICRBGKPDRHCR 8.8 Ki 4
CBLUNKVNKSMVMO 8.8 Ki 4
DOSWXEACORUGRU 8.8 Ki 5
HBYKTDPONPUZPO 8.8 Ki 7
NTCOZURJKJMLEZ 8.8 Ki 3
NTTOSPBYGRNOJQ 8.8 Ki 3
PQYKLGRHXIJMQB 8.8 Ki 3
QAESTHCUZJPQGF 8.8 Ki 9
WFSGQIXIGIQILN 8.8 Ki 4
DJGBDGBJUAFKHX 8.7 Ki 3
FREWUHPTJYJHEV 8.7 Ki 5
GNTLDZVFSGMZMM 8.7 Ki 3
GZKLJWGUPQBVJQ 8.7 pIC50 24 Yes
LVDRNYWTLKUNNT 8.7 Ki 4
OUDWCNZTASZGHL 8.7 Ki 5
PKEBCPIHEMJZIG 8.7 Ki 4
PNCPYILNMDWPEY 8.7 IC50 13
SGTFFUDLSDUTKM 8.7 Ki 4
UQMPYAUGLXZWSM 8.7 Ki 2
USIWFTPEBGPOSA 8.7 Ki 4
UYZCRXKULSDXTA 8.7 Ki 4
WLHRCQLHMHKOKG 8.7 pIC50 2 Yes
WPSYNFMKLRQHSU 8.7 Ki 3
JZHXLYHEWUWHQL 8.7 Ki 5
NXJYLDGTQWINTD 8.7 Ki 3
OZQHHXAYNRRVBN 8.7 Ki 7
PGMSQKAWALUURX 8.7 Ki 3
RJEWWPFKTYWTSS 8.7 Ki 6
CHKOUYJMMIYLHA 8.7 Ki 3
KYFDMTNYQFXNHE 8.7 IC50 2
LPAJCOGMIXSKKG 8.7 IC50 3
MVWVFYHBGMAFLY 8.7 pIC50 31 Yes
2D structure