Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
WIVOLWKUZIBRAF 9.0 pIC50 4 Yes
WJRKWJSQVYFSFK 9.0 Ki 5
XDIYJVCTGIMGBN 9.0 Ki 3
YPRBAEIXVWNGTP 9.0 Ki 3
LYVYZEAKTYROJI 8.9 Ki 4
VSWBSWWIRNCQIJ 8.9 Ki 23
KSCNWOYWUOCFLO 8.9 Ki 3
SCZDZQFTMOOIDO 8.9 Ki 6
ATBLUNCHMMWNHV 8.9 Ki 5
DSQXAOLERDQQCP 8.9 Ki 2
HYROFOKEXWNSCZ 8.9 Ki 2
IYHKQABMQSZQIQ 8.9 Ki 2
JVQZYMVBXVUIPJ 8.9 Ki 3
KBDQCTAMVLZQJL 8.9 Ki 4
MPEPNFOQCGMXGQ 8.9 Ki 5
OCDNDDLEORDHLQ 8.9 Ki 4
OXPSGDMBBBJERQ 8.9 Ki 4
QCNWWNZUDOKUHR 8.9 Ki 3
QYNUTROASKYRGA 8.9 Ki 3
SSVDRIUIQGHMLI 8.9 Ki 3
VSWBSWWIRNCQIJ 8.9 Ki 2
RHLJLALHBZGAFM 8.9 IC50 3
ZVZCHVBOZRWHPS 8.9 Ki 2
IJMJOPSALFMSMQ 8.9 Ki 3
UZNAGRGAFAEPBA 8.9 Ki 3
ZWJVFWQBNXKWES 8.9 Ki 4
AMDQVJAWEJXJFN 8.9 Ki 3
AVZNXYFYVNZTRE 8.9 Ki 2
CQABPCACTMBCQC 8.9 Ki 4
FSTGDSJHLKDASP 8.9 Ki 2
HWLHWHNTJPQILF 8.9 IC50 3
VZKPTHAFKKTYRC 8.9 Ki 4
WEZFJPKJUIGDPS 8.9 Ki 3
XAFOTAKURAOBIE 8.9 Ki 6
AOZOBKDTJZCKJE 8.9 Ki 4
CACGBSVXIXSELL 8.9 Ki 5
HSZTUDYUKZUFKK 8.9 Ki 3
WESSELXZMWZPLT 8.9 Ki 2
KAXNWVHHUKHNDK 8.8 pIC50 3 Yes
NHRXMVNDSUMAIN 8.8 Ki 3
SNEXCDCPPGPIOK 8.8 Ki 4
TZIDXYRBHBHFBV 8.8 Ki 3
UXYHEFDZIWONNI 8.8 Ki 3
VBMWRWYJANTSGH 8.8 Ki 3
XQDRWCFJBHLWPR 8.8 pIC50 8 Yes
IVMAVCHNIRPHMA 8.8 Ki 3
IDSYRZJPBIXBRS 8.8 Ki 2
BTYBILKFYYEYRM 8.8 Ki 6
KRIXMAGTZZHFLF 8.8 Ki 3
NAYUKRZMBPSGCB 8.8 Ki 4
2D structure