Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
XETGFITVYCWVGB 9.3 Ki 6
HETKYUVAGHVYTA 9.3 Ki 4
JOQJONDKZULBPP 9.2 Ki 4
UVEKKXRFQCNLQE 9.2 Ki 4
IENZQIKPVFGBNW 9.2 Ki 11 Yes
VPUVFWFLLOJNOU 9.2 Kd 2
CPWQIBJELMVKCH 9.2 Ki 3
DTQNYMCALLNMCV 9.2 Ki 3
FDRLNNNWCSSRPY 9.2 Ki 3
JMWBXYKHUPFCLZ 9.2 Ki 3
JWAHBXONODWUEH 9.2 Ki 3
HCKLMKILABOANU 9.2 Ki 4
KUSUAKLXHXASTN 9.2 Ki 3
LVCOTAHRPAKKNR 9.2 Ki 4
XLZHXAXXJVKTFM 9.2 Ki 3
DKZVZJLNJPUMKG 9.2 Ki 4
UUHRDARWBGSDJU 9.2 Ki 3
ASXGJMSKWNBENU 9.2 pIC50 12 Yes
IQRXOCGLSGCNLE 9.2 Ki 2
KWEAVTKRDHFTIH 9.2 Ki 3
SJDOMIRMMUGQQK 9.2 Ki 8
STMYXSKGGILJBE 9.2 Ki 2
FJIKITBGGGDJBY 9.2 Kd 3
RAPZEAPATHNIPO 9.2 pIC50 28 Yes
AADBHVDMLFAXQC 9.2 Ki 3
IIGHIMZENWTPRU 9.2 Ki 3
MGEPWLHHOOYNQU 9.2 Ki 3
PGWWSFHSBLBNGD 9.2 Ki 2
VITDWMDDGMNHHH 9.2 Ki 3
IMBDRGLQGCAYLF 9.1 Ki 4
QINUQIXOUYBPRY 9.1 Ki 4
GPVSQYKLAUEUBR 9.1 Ki 3
MCCWDRVXIBWEIB 9.1 Ki 3
PAUUPYPPPJQSIG 9.1 Ki 4
URHATDOBWHTBOV 9.1 Ki 2
ALXPTLNJYZORDB 9.1 Ki 3
AXOUSXBEKHBGLU 9.1 Ki 3
BXZWRAYRDLNDSN 9.1 Ki 3
DLMPCEBSXNLTAT 9.1 pIC50 5 Yes
GXZWKZAOGQRNTL 9.1 Ki 12
PKOIYURUOMCFSD 9.1 Ki 3
UJAZDXIAIGDQSX 9.1 Ki 3
PUSDBRIZNFZIFK 9.1 Ki 3
WYYRWPAVRAAIOL 9.1 Kd 3
ZPEIMTDSQAKGNT 9.1 Ki 35 Yes
CCJMGYBFMJJAIY 9.1 Ki 2
HCVFJHZVTICJEK 9.1 Ki 4
MMNXGMKPQQFESW 9.1 Ki 4
XPMVBFIBOSIETN 9.1 Ki 3
YCSBRVKGUOPSQB 9.1 Ki 2
2D structure