Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
CLADBLWFXVASRD 8.2 Ki 4
HEMORBXXFYODCC 8.2 Ki 3
NXJNUASOAQRPKJ 8.2 Ki 4
VCKUSRYTPJJLNI 8.2 Ki 6
YXYDEEZYQMLTIS 8.2 Ki 4
BVILLZIQPZNAQJ 8.2 Ki 3
LRLMUKKGKWCSTQ 8.2 Ki 4
MEKSQRMXWZHFIP 8.2 Ki 13
FKPDOXLGSMSHFA 8.2 Ki 3
FSAKTEBFSIPADS 8.2 Ki 2
HAISIGWLLOPIBJ 8.2 Kd 3
UZMKDOUDIGKWHV 8.2 Ki 3
IBNWNWKMISLVQT 8.2 Ki 8
IFVRVNMRXMDJCL 8.2 Ki 4
LEVRYVCMBBJQLU 8.2 pIC50 2 Yes
NSXHCXUYOMDHEJ 8.2 Ki 5
RVPGPLCUKORXKA 8.2 Ki 4
VHYJQKUBUIGDCY 8.2 Ki 3
WBCDPYPSNVABPM 8.2 Ki 3
DZTKYUPHGYMDEB 8.1 Ki 3
KVWDHTXUZHCGIO 8.1 pIC50 32 Yes
OWOQRXHVMOMTJK 8.1 Ki 4
ZKNQRQDTAWUUJL 8.1 Ki 4
GAWCPJXNKBSMOF 8.1 Ki 3
HGRPPZKIXIZLRX 8.1 Ki 7
IMKMRGOTDDUQHF 8.1 Kd 3
JKMSDGXSNFPBBL 8.1 Ki 2
CGCLDRKORPAFBZ 8.1 Ki 3
DZYBJTLUOQNDRI 8.1 IC50 3
PLDUPXSUYLZYBN 8.1 Ki 22
UHPXZGGJCMUMGZ 8.1 Ki 4
YNZFNGNFBKOQRH 8.1 Ki 4
ZUXABONWMNSFBN 8.1 Ki 29
BASQZMOJDHSJPS 8.1 Ki 4
BHUCMEWUSAGOPR 8.1 Ki 4
BTFVTAWVFBWGHC 8.1 Ki 4
BVRXELLJAMJMOD 8.1 Ki 4
DZVJBZTUTCHLSB 8.1 Ki 5
PPJRQXMDFSRWFH 8.1 Ki 3
QYNFZZOONQJAIB 8.1 Ki 3
RHTRBRRAADVASO 8.1 Ki 4
RNAQUCCCIRBEBB 8.1 Ki 6
SCPHBHCWLOVVMW 8.1 IC50 3
SDHKUGRGWQZRIK 8.1 Ki 3
WCGXKZZNDLNAMK 8.1 Ki 3
XJDCBRPORGPJTQ 8.1 Ki 4
YCKRBYBOMGAOET 8.1 Ki 2
YJWWBNSDIIFYRN 8.1 pIC50 6 Yes
PDAVXRWJDNCAQA 8.1 Ki 4
PXWNTBGUQKWMOQ 8.1 Ki 2
2D structure