Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
ZSBUPDFCHJYDDP 8.3 Ki 3
CPNQDPLKZHXMSB 8.3 Ki 6
NSXUBFCOCMDGJL 8.3 Ki 6
QQLBAAQRZXVWPZ 8.3 Ki 4
GDBMQKGUAQWBLZ 8.3 Ki 3
HAIKGHUWKLUYNG 8.3 Ki 2
IOEIAXGHDJMROV 8.3 Ki 2
KTBIQCRMHWZGGG 8.3 Ki 4
VZCKRSFEOTUZRB 8.3 Ki 3
GAFGMUJBSNDSHX 8.3 Ki 4
BKRGVLQUQGGVSM 8.3 Ki 18
FJHDZOUCRDBUGM 8.3 Ki 3
QAWYXANRFIWXDP 8.3 Ki 4
CQFKZCAKNRCPDY 8.2 Ki 3
KHXNVNNRQVTRJN 8.2 Ki 3
MMNXGMKPQQFESW 8.2 Ki 4
VZKPTHAFKKTYRC 8.2 Ki 4
LNEPOXFFQSENCJ 8.2 pIC50 33 Yes
RGGIGJAIAGZDRS 8.2 Ki 3
VQBXPTGVNAAIHI 8.2 Ki 7
XOZBPBSXMJMBOL 8.2 Ki 4
YIUMSISCOUIOHZ 8.2 Ki 7
YXGDGGYNHGGLOW 8.2 Ki 2
BAGJQDYWVPCFCU 8.2 Ki 8
HNTIGZIKHBPAFD 8.2 Ki 4
HRRBJVNMSRJFHQ 8.2 Ki 3
RORFUFVFDXKMOM 8.2 Ki 3
XIIKDAODIFECTH 8.2 Ki 6
GVOWTPVTYQMHDU 8.2 Ki 4
RZIZBETWVGIROJ 8.2 Ki 3
SHLHJQDYUNFBDK 8.2 Ki 4
SVLOMAHKFFJJIC 8.2 Ki 4
SXRUGRZXULZCBB 8.2 Ki 3
LGQDRXMJPKYZFZ 8.2 Ki 3
UVICRDSFJQQDJY 8.2 Ki 3
WDZOSSNSOBKEMP 8.2 Ki 4
FRUMSZUUBXPHHF 8.2 pIC50 4 Yes
HEEKUWDLPPDKMK 8.2 Ki 4
HJESDLDLPTXZBL 8.2 Ki 3
MGYNRIYGDOFIPG 8.2 IC50 3
OZUYIQYXHKJSCF 8.2 Ki 4
PANUNJICXXHAIL 8.2 Ki 4
QMMPFJGZOGDNHT 8.2 Ki 6
VFIDGXZRONKQBZ 8.2 Ki 5
WDDPQFVKUCBXKP 8.2 Ki 2
XEEZZVVUQHKGAE 8.2 Ki 2
POAIEWIIIXKJRN 8.2 Ki 4
QBFJWYVQWOPOQH 8.2 Ki 3
QVVUBPXTGZZTIW 8.2 Ki 2
YMCAXSPZJNPMHX 8.2 Ki 4
2D structure