Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
UNHGFWKSHHCRHF 8.4 Ki 3
LHLZWQUFUNHDHT 8.4 Ki 3
MFXXQERUKWXMIU 8.4 Ki 3
MNHTZNWGEQJHJN 8.4 Ki 3
OBGSISHOOKNBRI 8.4 Ki 2
PANBMHHKBRMYAL 8.4 Ki 5
PSQXMJPYXNSOJY 8.4 Ki 3
SDLAGDZFGDPJLC 8.4 Ki 2
FFXLCCZAXLBJFW 8.4 Ki 4
RHILFWFBQHFQIB 8.4 Ki 2
UIAXVFLURTXSJC 8.4 Ki 3
BERGTWZFNNPONR 8.4 Ki 3
LWIMUFCQSSEBRN 8.4 Ki 3
NJWKVUCAVMYELV 8.4 Ki 3
SOGVSTQOWIDIQK 8.4 IC50 3
CLKHJNVUYRXMGC 8.3 Ki 5
CQABPCACTMBCQC 8.3 Ki 4
GZYMKAZAURLMJX 8.3 Ki 3
KAHFZGUOPFFVHW 8.3 Ki 4
KCUCPEWBDAFYOT 8.3 Ki 3
LMLCPHRNHLEZIN 8.3 Ki 3
URKOMYMAXPYINW 8.3 pIC50 27 Yes
YMSCVVXGMWMEMM 8.3 Ki 6
DXKDPMJFFBCJSB 8.3 Ki 3
MRCKSWXOWOMYII 8.3 Ki 3
QOIHMWKAVCOQSF 8.3 IC50 2
VQLNHQYXLDPOCF 8.3 Ki 4
FBYRIOLLVVNZKA 8.3 pIC50 2 Yes
FPRCXYVVQHMAFI 8.3 Ki 3
OCBZSBUOYIQXSP 8.3 Ki 6
RCUUBRFHZZUGFH 8.3 Ki 5
CIMSZTVVTWKOJY 8.3 Ki 3
GHMHLQOFXXKCPZ 8.3 Ki 5
HNTIGZIKHBPAFD 8.3 Ki 4
HPKLBVVRBBCHTN 8.3 Ki 3
MKHBKMKCQKFQFC 8.3 Ki 3
RKHBPDFPBLQPEZ 8.3 IC50 3
SOUVKJLYRGDDOT 8.3 Ki 3
UHPXZGGJCMUMGZ 8.3 Ki 4
UTCOMQXMXQJEDA 8.3 Ki 5
KCWSSYYCEGZXTI 8.3 Ki 4
KTTHVCJSRNMDJY 8.3 Ki 3
ADSQCTGZHJXUFN 8.3 Ki 4
BQDGJNNXKPPHKX 8.3 Ki 3
CFECXSNWRXZHNR 8.3 Ki 3
IBAMCKKDXCRFQF 8.3 Ki 3
KLBQZWRITKRQQV 8.3 Ki 21
RMKWPAUMYJFUEG 8.3 Ki 4
XOZBPBSXMJMBOL 8.3 Ki 4
ZNFGZJGKELODLV 8.3 Ki 4
2D structure