Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
AEJCTJSNUNXYQL 8.5 Ki 4
BBIXFEYHANJCTO 8.5 Ki 4
BXERZGFRIILESM 8.5 Ki 4
KPTMOEWLVJTEEX 8.5 Ki 4
NFPVLBNNIZXLMJ 8.5 Ki 3
BYPMJBXPNZMNQD 8.5 Ki 18
HDOZVRUNCMBHFH 8.5 pIC50 26 Yes
IDZICZAULARHJJ 8.5 Ki 2
PTNLKWJYWYHWJE 8.5 Ki 3
RZKGYUBITDXCBT 8.5 Ki 3
BLFCXMMGSUUVCS 8.5 Ki 2
CKDALLRCYSNSRF 8.5 Ki 3
CKDALLRCYSNSRF 8.5 Ki 3
FPCCSQOGAWCVBH 8.5 Ki 16
IMBDRGLQGCAYLF 8.5 Ki 4
LASDMXNHWPCZMK 8.5 Ki 4
LGOXMVBGBCZVNL 8.5 Ki 3
WJFLJWNZAPQFEZ 8.5 Ki 3
ZFLJBXISNFUYBH 8.5 Ki 3
JOAHPSVPXZTVEP 8.4 Ki 19
DZEZXWSJRQPUTM 8.4 Ki 2
QGTFDZFDVRWNAC 8.4 Ki 2
UJELWGXJMXZTIC 8.4 Ki 3
XQPITIPYGHBCQW 8.4 Ki 3
HHXHWBGCTREPSZ 8.4 Ki 3
HVJHLWDXQXIFIC 8.4 Ki 3
JXZZEXZZKAWDSP 8.4 Ki 5
OALIYDQKZULGGT 8.4 Ki 2
SFTUKEODVLRSBF 8.4 IC50 3
CWRGETLEMMGBDH 8.4 Ki 3
DSMKEQAYQKRDDL 8.4 Ki 2
FTEANBXSHLNIRR 8.4 Ki 3
GENVWLSAPICTPF 8.4 Ki 3
LVDRNYWTLKUNNT 8.4 Ki 4
QQBCCUCHUBUQEQ 8.4 Ki 6
XRCQNHQVZIQOBE 8.4 Ki 4
XWUSTWDFKOHGNW 8.4 Ki 6
HBKDXPFFGLQBAS 8.4 Ki 3
OCDNDDLEORDHLQ 8.4 Ki 4
QPJSKVVDVIYOKV 8.4 Ki 3
XOZFOKIHXFIGLO 8.4 Ki 7
AGNYFINNIVFBHA 8.4 Ki 4
BRSPJIFNHOLFQU 8.4 IC50 3
GRHNWNVQLGTXTE 8.4 Ki 3
LXGZSTDLYCGLAE 8.4 Ki 4
MDXDUERQAFAILI 8.4 Ki 5
PPAIEDLGYFCKEB 8.4 Ki 4
XGXYGEYUGTVZAR 8.4 Ki 6
ZFZUYTCCHMWWTD 8.4 Ki 9
KEFRGKGZIBGWEZ 8.4 Ki 4
2D structure