Target Details
UniProt ACP35348
Gene SymbolADRA1A
Protein NameAlpha-1A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,709
  • Clinical molecules 128
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (1,709)
InChIKey pChEMBL Type Targets Clinical
QORSFUXHRJFURF 11.0 Ki 3
JCWKQYAUPMXURC 10.7 Ki 3
ANZIISNSHPKVRV 10.4 Ki 3
NJLNPETVWRAQNN 10.4 Ki 3
DASDCIRXSWKVTA 10.3 Ki 4
JCWKQYAUPMXURC 10.3 Ki 3
AACTUBFOGVFADC 10.2 Ki 3
ARVUOFMRSSPQPL 10.2 Ki 3
MMJIOQBMUWSARZ 10.2 Ki 3
LOSOVXONSYGDJN 10.2 Ki 3
VGCCDDCHXNJOMD 10.2 Ki 3
LKCYPDONQAJLQQ 10.2 Ki 3
KFFBTOAYJRDMAT 10.2 Ki 3
OZLVILGCRABIEJ 10.2 Ki 3
GUROZSUTVHXVSF 10.1 Ki 3
JGLLHUJRQIQLNY 10.1 Ki 4
OTPCOGQCPMOGMX 10.0 Ki 4
AECCHTQUIJEKGQ 10.0 Ki 5
DFCWYIOPOZJPPQ 10.0 Ki 3
FBYRIOLLVVNZKA 10.0 pIC50 2 Yes
FOMUZVDWSAHVBW 10.0 Ki 3
FXFOLWSUKNFCFK 10.0 Ki 3
GUCRUSFOVGPMOS 10.0 Ki 5
JHAYORQLJMSTOO 10.0 Ki 3
JICRZQUVMVWMQI 10.0 Ki 3
JXDBPRQKWGFDFQ 10.0 Ki 3
LUKZCSDJGOLWJZ 10.0 Ki 3
MQRCKTYDHDXFKE 10.0 Ki 3
NPUFUXHUZGWJII 10.0 Ki 5
UIJPUNVNCOWEMQ 10.0 Ki 3
VKJWHZVTJUKYAU 10.0 Ki 3
VRERDSWPFMZSEX 10.0 Ki 3
VWLOQZCQYQZEHT 10.0 Ki 3
ZTAFSHDVHGVXTJ 10.0 Ki 3
MVYCXEXQTMBCNB 10.0 Ki 3
DMMNMIJPRNMLBQ 9.9 Ki 3
LDXAPIWITLZXNM 9.9 Ki 3
UYWFSEXEAMKGLC 9.9 Ki 3
ZZNMPZNCGBNJBR 9.9 Ki 3
GSTGFHBCLUCUEI 9.9 Ki 3
USHDDUDLXIGXFA 9.9 Ki 3
ZRWCHZNUZHLTHH 9.9 Ki 3
ZCVMWBYGMWKGHF 9.9 pIC50 19 Yes
CHSVWGZALFVOMB 9.8 Ki 3
KQUFPVZMSZOANN 9.8 Ki 3
QWLYOONHUJJIHC 9.8 Ki 3
RMKDNMUUFMLYDR 9.8 Ki 3
AROSMOXZDJFPHJ 9.8 Kd 2
CBACROBVDLICEW 9.8 Ki 3
CSXUKDQJFRHATO 9.8 Ki 2
2D structure