Target Details
| UniProt AC | P34998 |
|---|---|
| Gene Symbol | CRHR1 |
| Protein Name | Corticotropin-releasing factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 35
- Clinical molecules 0
- Avg pChEMBL 8.13
KEGG Pathways (5)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BIIOOWPFSOAZSO
|
10.2 | IC50 | 2 | — | |
BXTRKRJIYZENAK
|
9.6 | IC50 | 2 | — | |
HPYIIXJJVYSMCV
|
9.1 | IC50 | 2 | — | |
KFUIXDNQSMKKJQ
|
9.1 | Ki | 2 | — | |
GYHCTFXIZSNGJT
|
9.1 | Ki | 4 | — | |
PNMZQWKBJIQQJL
|
9.0 | IC50 | 2 | — | |
YIHRBRJTFIGRRV
|
9.0 | Ki | 2 | — | |
YIHRBRJTFIGRRV
|
9.0 | Ki | 2 | — | |
KBXXQHLYNYCQAE
|
8.7 | IC50 | 2 | — | |
UPVFHCQGPPALAB
|
8.5 | IC50 | 2 | — | |
BIIOOWPFSOAZSO
|
8.4 | Ki | 2 | — | |
GBONBLHJMVUBSJ
|
8.3 | Ki | 2 | — | |
GBONBLHJMVUBSJ
|
8.3 | Ki | 2 | — | |
ZXQWGXPBQWFYKG
|
8.2 | IC50 | 2 | — | |
QEEJLLNYQOBRRM
|
8.2 | Ki | 2 | — | |
FUFHRWPFPLHLRL
|
8.1 | Ki | 2 | — | |
QEEJLLNYQOBRRM
|
8.1 | Ki | 2 | — | |
BBNGUKKQYPAMTB
|
8.1 | IC50 | 2 | — | |
BPJKLNRBFUIHRZ
|
8.1 | IC50 | 2 | — | |
CMZOBLKSINEYCW
|
8.0 | IC50 | 2 | — | |
IMAXYSCPKOIFBE
|
7.9 | IC50 | 2 | — | |
WBNJZEUGPLZJAS
|
7.9 | IC50 | 2 | — | |
HBBPLUNKEXJZQZ
|
7.8 | IC50 | 2 | — | |
KCPHVCVRMSDLQN
|
7.8 | IC50 | 2 | — | |
LSFVOPLRJHUUNQ
|
7.8 | IC50 | 2 | — | |
QBZAHNFIFYKUAQ
|
7.7 | IC50 | 2 | — | |
YZGWWUVHEOPLKF
|
7.6 | IC50 | 2 | — | |
BYXIIQICFOHBMN
|
7.5 | IC50 | 2 | — | |
DOEWJZPYNWPPDF
|
7.5 | IC50 | 2 | — | |
FFMNQLRIMQJKNK
|
7.4 | IC50 | 2 | — | |
ZEGBRYNTIJDVHP
|
7.4 | IC50 | 2 | — | |
IQJNGBXKROFQRM
|
7.3 | IC50 | 2 | — | |
QBKRBQAPESJEEH
|
6.9 | IC50 | 2 | — | |
BTXNYTINYBABQR
|
6.5 | IC50 | 2 | — | |
VHTUCYOJWFRPJN
|
6.3 | IC50 | 2 | — |