Target Details
UniProt ACP34995
Gene SymbolPTGER1
Protein NameProstaglandin E2 receptor EP1 subtype
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 47
  • Clinical molecules 0
  • Avg pChEMBL 7.35
Top Co-occurrence Targets
Active Molecules (47)
InChIKey pChEMBL Type Targets Clinical
HQNOTLSNWDHOJY 9.1 IC50 3
VTRCWWBWFOAGSU 9.1 IC50 2
MJUSLUQFEHEIHA 8.8 IC50 2
FECWOVCONGPURJ 8.8 IC50 3
ZOQXTNLUBHPZOZ 8.7 Ki 5
RRDVGFBNUNMAKI 8.4 Ki 2
MRBWBFJXHIUJNQ 8.4 Ki 2
JCCQFQOPADDTRS 8.3 Ki 2
YVTIVJFGJQZENO 8.3 Ki 4
KWCSGHGCXOSYQY 8.3 IC50 3
KMTAAGONUZDGDG 8.2 IC50 3
HJPAXYLYYQIFCK 8.1 IC50 2
XEYBRNLFEZDVAW 8.0 Ki 7
CQBVTZDISUKDSX 8.0 Kd 4
CBDBSQHFOYMVSD 8.0 Ki 3
HIFJCPQKFCZDDL 8.0 Ki 5
IILDGMMYAPPHGT 7.9 Ki 2
RVMVCPKCWWFOEL 7.8 IC50 2
ONFDZOUFCUXZFV 7.8 Ki 2
YIJWSWGNFRVEHD 7.7 IC50 2
XZFRIPGNUQRGPI 7.6 Ki 7
UYYILQXGACUYJD 7.5 IC50 2
FAPQZCFUFGJPFI 7.4 IC50 4
CZCMZYYRRYEIHW 7.4 Ki 2
PNVFGVWWQZJNKR 7.2 Ki 2
SXDFNJNZJPSKSR 7.2 Ki 2
PTOJVMZPWPAXER 7.1 Ki 3
XNLHIHZVDIHXJA 7.1 Ki 2
UQZVCDCIMBLVNR 7.0 Ki 3
VCZASWFGPQFOFT 6.8 Ki 2
FHQODQOFYNUYNU 6.6 Ki 3
AJGJMWUDDSWHOG 6.6 Ki 2
PXGPLTODNUVGFL 6.5 IC50 4
KVSPDLWJCJFYEZ 6.5 Ki 3
HIZNWXUSWJBZEM 6.4 IC50 2
YTZPMGSDIYCPCW 6.4 IC50 2
NZGFSDWJUZOAAX 6.4 Ki 6
VJYUXEQWPPXOLL 6.3 IC50 2
VJGGHXVGBSZVMZ 6.3 IC50 3
BHGLRNRVCYDAJB 6.3 IC50 2
PXGPLTODNUVGFL 6.3 Ki 7
VJGGHXVGBSZVMZ 6.2 IC50 3
ZELKHLBDQHQEJW 6.2 IC50 2
CCIGYTQGGWYUNA 6.2 IC50 2
HMHNXLVVOUOPHR 6.1 IC50 3
WRTHARKMYHJTNQ 6.1 Ki 3
CHDOVUGJRCWTAC 6.0 IC50 2
2D structure