Target Details
| UniProt AC | P34947 |
|---|---|
| Gene Symbol | GRK5 |
| Protein Name | G protein-coupled receptor kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 71
- Clinical molecules 8
- Avg pChEMBL 6.38
KEGG Pathways (3)
Active Molecules (71)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HHFBDROWDBDFBR
|
6.0 | Ki | 40 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JRLSUZIPUYDUKX
|
6.0 | Ki | 22 | — | |
KDKUVYLMPJIGKA
|
6.0 | Ki | 91 | Yes | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KWGIZLMNJXFPFV
|
6.0 | Ki | 3 | — | |
LHAZDFBNDIQNSG
|
6.0 | Ki | 4 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NDSSSMYGJDDEPB
|
6.0 | Ki | 3 | — | |
OWRXHGAFWZFFCW
|
6.0 | Ki | 113 | — | |
PDXVRCZNPFLZJP
|
6.0 | Ki | 3 | — | |
PWMGIYOLYSEHBN
|
6.0 | Ki | 3 | — | |
QDNSHFHBLOTJEL
|
6.0 | Ki | 3 | — | |
RPBKUXXUYPWIPS
|
6.0 | Ki | 3 | — | |
SGPKBJQYKUQGKV
|
6.0 | Ki | 3 | — | |
SJLQDZDKTVBBLP
|
6.0 | Ki | 9 | — | |
UIRCQOKSJDLYBB
|
6.0 | Ki | 50 | — | |
VRKITNLDCQGIJI
|
6.0 | Ki | 3 | — | |
XTVULKIROSNNTG
|
6.0 | Ki | 29 | — | |
YKLNVZIGQDKBKJ
|
6.0 | Ki | 3 | — | |
ZXYUSNLUAQYJFK
|
6.0 | Ki | 3 | — |