Target Details
| UniProt AC | P34947 |
|---|---|
| Gene Symbol | GRK5 |
| Protein Name | G protein-coupled receptor kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 71
- Clinical molecules 8
- Avg pChEMBL 6.38
KEGG Pathways (3)
Active Molecules (71)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ACLLLJSNOCYQOJ
|
7.9 | IC50 | 8 | — | |
HKSZLNNOFSGOKW
|
7.6 | Ki | 118 | — | |
GYMOXCZIQHPXOH
|
7.6 | IC50 | 6 | — | |
NWMPVMMGSHXANZ
|
7.4 | Ki | 58 | — | |
PTJBMQVUHYZJLN
|
7.3 | IC50 | 5 | — | |
MWVKLRSIDOXBSE
|
7.2 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
AEYLJTAIDDIOBA
|
7.1 | Ki | 53 | — | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
FENQBUSSSWWVGH
|
7.0 | Ki | 3 | — | |
SKZTUPIPRLPDKY
|
7.0 | Ki | 3 | — | |
POEIXYXZODKFHQ
|
6.8 | IC50 | 2 | — | |
XYUFCXJZFZPEJD
|
6.8 | IC50 | 23 | Yes | |
ZGDYBJXDIXVTLV
|
6.8 | Ki | 54 | — | |
VHISWSDHEWXRKH
|
6.7 | IC50 | 2 | — | |
URNZTLZSAVLTIZ
|
6.7 | Ki | 26 | — | |
ILFWAZIPGQKPSC
|
6.7 | IC50 | 3 | — | |
HJYHJYGXRBYDIG
|
6.6 | Ki | 23 | — | |
WAKGEHXTOOFEAE
|
6.6 | Ki | 27 | — | |
SRDLWBLWLYRNNX
|
6.6 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.5 | Ki | 231 | Yes | |
BLMBNKDQXGINRE
|
6.4 | IC50 | 3 | — | |
XBRPSBXARPNOBH
|
6.4 | IC50 | 2 | — | |
LUPCHAFIKZSOOK
|
6.4 | Ki | 15 | — | |
VNDWQCSOSCCWIP
|
6.4 | Ki | 39 | Yes | |
XZWVOUQIYLZUCJ
|
6.4 | Ki | 23 | — | |
ZGZVRPRSFXRGCF
|
6.4 | Ki | 76 | — | |
SDBOIBYRBWPIEL
|
6.3 | Ki | 31 | — | |
WHVFDYQCAMPLMS
|
6.3 | Ki | 20 | Yes | |
LZZDXJOCYMXGCD
|
6.3 | IC50 | 2 | — | |
XWCWGOOBIPAWPA
|
6.3 | IC50 | 2 | — | |
DWTNLZZEPSCAIH
|
6.2 | Ki | 25 | — | |
HFNKQEVNSGCOJV
|
6.2 | Ki | 18 | — | |
OAVGBZOFDPFGPJ
|
6.2 | Ki | 42 | Yes | |
QVNZKVACBBTKSL
|
6.2 | Ki | 38 | — | |
RYYNGWLOYLRZLK
|
6.2 | Ki | 104 | — | |
WDARYLSSWBWVCU
|
6.2 | Ki | 49 | — | |
XUFLBSMTYMFOQH
|
6.2 | Ki | 43 | — | |
XMPOFQWNHXAUKI
|
6.2 | IC50 | 2 | — | |
RDEKYROQCDTNPC
|
6.2 | IC50 | 2 | — | |
BXTYCBBDHNQJNG
|
6.1 | IC50 | 3 | — | |
GZAQDFYUURXJSL
|
6.1 | Ki | 8 | — | |
HZPACYSNLOCDLW
|
6.1 | Ki | 48 | — | |
JMIIFJIJWDCOEP
|
6.1 | Ki | 15 | — | |
UOVCGJXDGOGOCZ
|
6.1 | Ki | 59 | — | |
VETBKPDTHQZBKH
|
6.1 | Ki | 3 | — | |
WINHZLLDWRZWRT
|
6.1 | IC50 | 201 | Yes | |
QHJAGBLQKDHNBD
|
6.1 | IC50 | 2 | — | |
ZGIZCVACDOOTHQ
|
6.1 | IC50 | 2 | — | |
AQKQATGZIKRZMQ
|
6.0 | Ki | 16 | — |