Target Details
UniProt ACP34903
Gene SymbolGABRA3
Protein NameGamma-aminobutyric acid receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,007
  • Clinical molecules 0
  • Avg pChEMBL 7.68
Top Co-occurrence Targets
Active Molecules (1,007)
InChIKey pChEMBL Type Targets Clinical
PHYVZWNIDCNYML 8.2 Ki 2
QVOYXYWXOMVGNY 8.2 Ki 4
ACUNYYFYYWOKOD 8.2 IC50 16
NKSBSXBZWIZUKS 8.2 Ki 3
IPEQYLWHCRAOTC 8.2 Ki 6
QAMANTJYKWSLNP 8.2 Ki 6
XUJMJGTVTZESCM 8.2 Ki 7
YUOOYQDBXTWPKL 8.2 Ki 16
DKGPQXLYULZUKP 8.2 Ki 2
HGJUDXDUSGEVOX 8.2 Ki 6
AZIRFKLEFANUIC 8.2 Ki 6
CNFLHWVYIFARIM 8.2 Ki 7
OTQXKRRISJPTFS 8.2 IC50 16
RLFKILXOLJVUNF 8.2 Ki 16
VUSVWZBQTTWZGJ 8.2 Ki 5
WMCJJXHYPNOCMT 8.2 IC50 16
ZRPUPUBWCXFOCY 8.2 Ki 16
KVQODEJTLJVMEH 8.1 Ki 4
LDRJMZJUSNJPQM 8.1 Ki 2
UOYBEURVYWDNBS 8.1 Ki 5
WQYYZNGOTUCWQX 8.1 Ki 5
QCNXINIQJHEAHO 8.1 Ki 4
QNLKJSGZMGMFBW 8.1 Ki 6
RJOMRLSAWXNFSU 8.1 Ki 4
BGOCUVAKPSPUAI 8.1 Ki 2
MZTRNWROWIGTRB 8.1 Ki 7
NMIWQCPJXNFYRR 8.1 Ki 5
VIILRVHOGYZXSZ 8.1 Ki 2
XRAXGFWJSVWBHB 8.1 Ki 4
ZAKVPALBELHKFH 8.1 Ki 6
DKCAUMRZSZVJCP 8.1 Ki 16
HNKGGOINWLAPIU 8.1 Ki 4
IVGTVZGLPHBTJV 8.1 IC50 16
IVGTVZGLPHBTJV 8.1 IC50 16
QIZPCEVRKTWHIE 8.1 IC50 16
QVIQGNJPFOVZBZ 8.1 Ki 16
YHNNMZUUFMJQQY 8.1 IC50 16
ZACQJMKEQBFUDN 8.1 Ki 6
IBIAGNJTCFFVTB 8.1 Ki 5
YMEKUDZYTKIXGP 8.1 Ki 2
GAMSSMTVVVDEJR 8.1 Ki 4
HEGJYRQUDMITRQ 8.1 Ki 6
PYXJKYJAFMLYMS 8.1 Ki 6
PZIQTZQOFYKORR 8.1 Ki 6
INJKUEAWCDOGAY 8.1 Ki 3
LLJUUCOIBTZXIJ 8.1 Ki 6
UWQBBGFHDXOYNN 8.1 Ki 2
MLRKAMHWRLRODO 8.1 Ki 4
XGJLRKVQXMSBJW 8.1 IC50 16
IXGIOXIKQZCZIK 8.0 Ki 8
2D structure