Target Details
UniProt ACP34903
Gene SymbolGABRA3
Protein NameGamma-aminobutyric acid receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,007
  • Clinical molecules 0
  • Avg pChEMBL 7.68
Top Co-occurrence Targets
Active Molecules (1,007)
InChIKey pChEMBL Type Targets Clinical
AOZALWRGTMILIK 8.3 Ki 6
PFJHXYJLEIZLGQ 8.3 Ki 6
PPTYJKAXVCCBDU 8.3 Ki 7
SSJXJXJUHUAOQL 8.3 Ki 6
GTLAYADJMQDCQJ 8.3 Ki 5
KCWCNDXYAPQOHU 8.3 Ki 5
QQIVOICVQUEJEG 8.3 Ki 4
YGKSPOBIXHTPMV 8.3 IC50 16
YLPHFEFMBAMSKS 8.3 Ki 5
ZKVGHURGXXUFQB 8.3 Ki 6
ACMQMUZDLQDWTK 8.3 Ki 16
AHHSTGLUTRNWRJ 8.3 Ki 6
ASOMQCZKXCZAAQ 8.3 Ki 2
CLKDKLQSBMZIQH 8.3 Ki 2
GOCZPCXRIJMRNR 8.3 Ki 16
PHOATQSOBKATTD 8.3 Ki 16
PTRXPVDOTUGGHW 8.3 IC50 16
UKHFPVCOXBJPIN 8.3 Ki 17
XQXFLYIUHYKDHV 8.3 Ki 4
BGRWSFIQQPVEML 8.3 Ki 6
SOLFHEZOCDBPSQ 8.3 Ki 4
VAJLZGPUVKNCRO 8.3 Ki 6
FBBGZDOIPFFHLI 8.3 Ki 4
JXUDSFIVAUVTDY 8.3 Ki 2
LRHBSPDBIHZAOV 8.3 Ki 2
MSYBIYCNXBCGOA 8.3 Ki 2
ZWWZTFYQCITUTK 8.3 IC50 16
BEUFUKHUURWENE 8.2 Ki 4
CFMPKKXOXYNZHF 8.2 Ki 6
MNTGRSPARUFALM 8.2 Ki 5
KOVRZNUMIKACTB 8.2 Ki 17
QWWODAPIEHJFQG 8.2 Ki 16
ZGEGOFCLSWVVKG 8.2 Ki 5
ALBKMJDFBZVHAK 8.2 Ki 16
BTLWEEGNXUJKKB 8.2 IC50 16
KIVQXKXZISOGBE 8.2 Ki 17
KXZNTMNIMNTHIP 8.2 Ki 2
NKIYALPHXLYICR 8.2 IC50 16
VCPRTCGXKBSFJJ 8.2 Ki 4
YUSWMAULDXZHPY 8.2 Ki 20
ZRRVSALMQDOQAX 8.2 Ki 16
MRBNIDFDWVVALT 8.2 Ki 5
RTRIMAMBTITPNP 8.2 Ki 6
YZRXMMCBUVDBFF 8.2 Ki 6
ZJQHPWUVQPJPQT 8.2 Ki 17
ZLTZGADBISMZKB 8.2 Ki 4
BDISWVKOOATATE 8.2 Ki 16
DNSPBVIIBSAYPW 8.2 Ki 5
DTUMUPWQPZERNQ 8.2 Ki 2
JHXTWTGOXRMYJM 8.2 Ki 3
2D structure