Target Details
UniProt ACP34903
Gene SymbolGABRA3
Protein NameGamma-aminobutyric acid receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,007
  • Clinical molecules 0
  • Avg pChEMBL 7.68
Top Co-occurrence Targets
Active Molecules (1,007)
InChIKey pChEMBL Type Targets Clinical
AHTXTFPELOVMKB 8.8 Ki 6
BCEWAHBYIZQWJY 8.8 Ki 5
CMRJVDJLBFKXKL 8.8 Ki 4
KSYVJHGNJMYDIQ 8.8 Ki 6
MFZNONRIQYSLMZ 8.8 Ki 6
OJLYUGSSUKAWJC 8.8 Ki 16
XGMPKZHPHLEVGE 8.8 Ki 4
KKWDMTXJUXKNOU 8.8 Ki 7
KVKYGVOAHGNAKZ 8.7 IC50 16
OIVNHVRINWMDTH 8.7 Ki 5
PCZLQMGFNUNVOM 8.7 Ki 6
KVQKVRWATUWLAO 8.7 Ki 5
LOZNAQDBHKVLRN 8.7 Ki 6
IHDXFSAXAJRBOG 8.7 Ki 5
DLGWSCNXWHDMHZ 8.7 Ki 4
FTBGMXWQYKNAKT 8.7 Ki 6
IPBXYXQZSUGQTK 8.7 Ki 5
KVTRKSLNWMZSSN 8.7 Ki 4
RFOXASLOAHSVQO 8.7 Ki 3
YKKWBLSUYZOORV 8.7 Ki 6
PUNLHXOQDSEUQP 8.7 Ki 4
QTEUJQNPMLXVLL 8.7 IC50 16
WRXDVVALWQGPMW 8.7 Ki 16
ZAYUCIMDULREJZ 8.7 Ki 4
BKIXSCDBYYIHQI 8.7 Ki 5
QCILNSKJADMOQI 8.7 Ki 4
BWWQXKSOWUMHAQ 8.6 Ki 6
JOHKRJNYKDHTID 8.6 Ki 6
SJAGJFDQMIAULO 8.6 Ki 6
ZOCSXAVNDGMNBV 8.6 IC50 16
VJVAWKPXJCDEQG 8.6 IC50 16
HJNOESUOZGNLKO 8.6 Ki 6
OJVFFZLXISLIFZ 8.6 Ki 6
OKGJPMZATLJSGV 8.6 Ki 6
WZNQGAWPCOPXOK 8.6 Ki 4
XPSAGIQSESMIJK 8.6 Ki 6
DZPQKPSHACGLKC 8.6 Ki 6
GXKGSEUULCEOTM 8.6 Ki 5
IGTNDWINIZAURX 8.6 Ki 3
KYKSBUKRCPZJCX 8.6 Ki 4
FFIJKSHMFVHCAE 8.6 Ki 3
YCTZWWGYTRDQQM 8.6 Ki 3
QSEBFHRZNPGODU 8.6 Ki 6
CHIFCDOIPRCHCF 8.6 IC50 16
CHQPOBHNDRMXFK 8.6 Ki 18
DKSWXNFPYZCJFU 8.6 Ki 6
STHRYAZDXIDVJO 8.6 Ki 6
OXRXBJGSNZVEPW 8.5 Ki 4
CBKOOGJFEQBENF 8.5 Ki 4
KVKYGVOAHGNAKZ 8.5 IC50 17
2D structure