Target Details
UniProt ACP34903
Gene SymbolGABRA3
Protein NameGamma-aminobutyric acid receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,007
  • Clinical molecules 0
  • Avg pChEMBL 7.68
Top Co-occurrence Targets
Active Molecules (1,007)
InChIKey pChEMBL Type Targets Clinical
WGRVAGIQTHEEQW 9.0 IC50 16
YLDRVNNGBACDSD 9.0 Ki 6
BSBLYLUAUVTSMM 9.0 IC50 16
GSLDBWNPXFIQAV 9.0 Ki 2
HNGRWUCKESPKRC 9.0 Ki 6
LSVOXYMZIGSSNB 9.0 Ki 6
LYXHWNNDUVMWRX 9.0 Ki 3
PTTQXDBPTFOCMT 9.0 Ki 6
UFTKNTUWDMJOIX 9.0 Ki 16
VNSQMHJPVJKTNQ 9.0 Ki 3
LICVBNQRZFPUHS 8.9 Ki 4
MTNLFTKJHWYWQV 8.9 Ki 4
OWOWBGNEZCVQKU 8.9 Ki 2
PELQRWYXKWRIDE 8.9 Ki 2
JAOIJSLHKQEWQB 8.9 Ki 4
LHMYCKKRCBXCBI 8.9 Ki 5
NPISRJOTBMWCDJ 8.9 Ki 2
QTYHDQOTKBKPBQ 8.9 Ki 3
SEWXZWMBVGJJPG 8.9 Ki 7
VJMXGRAYTDRKAO 8.9 Ki 6
ISZRIZPRXUQOMU 8.9 Ki 5
AWOOMIRCBITDFK 8.9 Ki 6
BJYKRVMKNGJKKZ 8.9 Ki 6
HOQUSTXYXSUJDG 8.9 Ki 6
JGVFVEUZTKIPIB 8.9 Ki 2
KYDURMHFWXCKMW 8.9 Ki 6
LWUDDYHYYNNIQI 8.9 Ki 6
OGBTVLIUFUJHTH 8.9 Ki 5
SGQQJEBYGVTMRA 8.9 Ki 3
DGBIGWXXNGSACT 8.9 Ki 16
RLLAIMNJXRQPNZ 8.9 Ki 2
BGVDDMWFMIAGGF 8.8 Ki 5
IYYLIZWRYYVEPH 8.8 Ki 4
JOFWLTCLBGQGBO 8.8 Ki 8
VREFGVBLTWBCJP 8.8 Ki 7
WXEWBVGLBRURRV 8.8 Ki 3
YTGZSWOWFGVAFH 8.8 Ki 7
ZQLPLWRQUVVKJZ 8.8 Ki 6
WQCOYHWSQLUYIH 8.8 Ki 3
UIBMSUDAMPUYHS 8.8 Ki 2
IUHKSTINHDUYRO 8.8 IC50 16
JJGMNYOOQJMINL 8.8 Ki 3
QBYZDDIMNITMSB 8.8 Ki 6
QGMKNRLNMKUUEC 8.8 Ki 2
SBVOTVOGQYZEOU 8.8 Ki 3
SSTBAKDUFHYWMX 8.8 Ki 2
XTZAPIKNFFKUDJ 8.8 Ki 2
HEFBZEKZYFOEGG 8.8 Ki 2
LLHQBHOWDZNCNK 8.8 Ki 5
MKQJGNJLLCPKEB 8.8 Ki 2
2D structure