Target Details
UniProt ACP34903
Gene SymbolGABRA3
Protein NameGamma-aminobutyric acid receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,007
  • Clinical molecules 0
  • Avg pChEMBL 7.68
Top Co-occurrence Targets
Active Molecules (1,007)
InChIKey pChEMBL Type Targets Clinical
WDBBCFFNOHDOBT 9.2 Ki 5
BLJPKQXXDFIIFR 9.2 IC50 16
BUTCFAZTKZDYCN 9.2 Ki 6
XJMIBNLJFYSGAR 9.2 IC50 16
LYZCPNJIFQNJQM 9.2 Ki 3
MTOXGGJOEHOEJT 9.2 Ki 5
NZMJFRXKGUCYNP 9.2 Ki 6
UZZBNSRTLAFTLY 9.2 Ki 2
VQOOIUSVMMFXEJ 9.2 Ki 4
VXVLSQVFRWSMKF 9.2 Ki 6
DSDYDTCIWBGXBT 9.2 Ki 2
GTPDUXMCZZEOBE 9.2 Ki 4
KMGQMDWTLIZLHG 9.2 Ki 4
BQDUNOMMYOKHEP 9.2 Ki 6
FNCCIRFBYGUBRQ 9.2 Ki 5
FYOXWZFDOADHOW 9.2 Ki 6
OLKUNPKISSHQBO 9.2 Ki 6
QVMKXYFWXJHPIX 9.2 Ki 2
QZDWWRKBDPYMIP 9.2 Ki 6
RGDHMJMNRYQXCW 9.2 Ki 6
RWUOGVWORJUNJA 9.2 Ki 4
YWVNAIWRDXBOOS 9.2 Ki 6
XXRKXVKJMSIZSM 9.1 Ki 6
JLCBYDSLJHLQQB 9.1 Ki 5
GMDXFYPWVIKBFF 9.1 Ki 4
QYSYOGCIDRANAR 9.1 Ki 7
JFGUJXZLJIUVPZ 9.1 IC50 16
JNJUWXAKLRKXII 9.1 Ki 6
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
VZKRZUPJCVFVGR 9.1 IC50 16
BJDIHPUUUSHMRK 9.1 Ki 2
LODWVHSNNGQTKI 9.1 Ki 3
ZPSBXQBYCQOCEU 9.1 Ki 6
QIWRIQRYIRGJCG 9.1 Ki 4
FAEJWVCMADNLAQ 9.1 Ki 4
MPEKCHDBHNYAJG 9.1 Ki 2
RYKBQSSZEXHGJL 9.1 Ki 5
UJBOQYCZTOTBAN 9.1 Ki 4
YJZGQBGGTBIAOP 9.1 IC50 16
GPTKIASBZUGFEQ 9.0 Ki 3
PNEOQFYBCKZRBL 9.0 Ki 3
VXSLAFXNESWHFV 9.0 Ki 2
AQKFCEWRKDXGMK 9.0 Ki 16
BYMDBFGHCDTBMT 9.0 IC50 16
CHMFFBQMSYJXTP 9.0 Ki 6
IPHSQMSRIWZULE 9.0 Ki 16
KDMMIKQMHNBKAV 9.0 Ki 17
OFBIFZUFASYYRE 9.0 Ki 16
RZOFEWOHNOOHND 9.0 Ki 6
2D structure