Target Details
UniProt ACP34903
Gene SymbolGABRA3
Protein NameGamma-aminobutyric acid receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,007
  • Clinical molecules 0
  • Avg pChEMBL 7.68
Top Co-occurrence Targets
Active Molecules (1,007)
InChIKey pChEMBL Type Targets Clinical
JWODBROOGAIDRT 10.0 Ki 3
ORCNDQDLFHQBRB 10.0 Ki 3
KWBJTSIHFVATSO 10.0 Ki 3
CGMJQQJSWIRRRL 9.9 Ki 6
CUCYVGNNTAIIAN 9.8 Ki 4
OWENCIOAIROJMF 9.8 Ki 3
MZFKWSFOAVBLQM 9.8 IC50 16
VACJUKKURQMWHE 9.8 Ki 5
UAISVGZOWWUBIG 9.7 Ki 2
LNPVVDKIXXYELR 9.7 Ki 3
LWUDDYHYYNNIQI 9.7 Ki 7
WFPXOWCKXUEKCA 9.7 IC50 16
YMMRGIIZANFGIG 9.7 Ki 6
GOIFCXRIFSYPFG 9.7 Ki 5
QUUNMICPMYIHFS 9.7 IC50 16
UWXAQZGCSSYTJL 9.7 Ki 6
KVKWRJDNIJTMGN 9.6 IC50 16
QKIWQBLNTSQOLY 9.6 Ki 6
IQKMZIHHJYCEKH 9.6 Ki 5
JUNLOSOXNSBSNV 9.6 Ki 3
ZRKDDZBVSZLOFS 9.6 Ki 6
FIXFKUDATBTRAZ 9.5 Ki 4
VYBPWFTWAKMZPZ 9.5 Ki 5
CMSKDYKEKYIJSD 9.5 Ki 5
NVETZYIXXYETLA 9.5 Ki 6
KWZFUKSTRXYXTQ 9.4 Ki 3
NURMFSYNABAOFU 9.4 Ki 6
PEBWTLIJBCZFOA 9.4 Ki 6
RUOVJURXWIHZPL 9.4 Ki 5
AJWPZYMLAILYCO 9.4 Ki 5
LCDOZBPYZHDFGO 9.4 Ki 5
NTQIDFIQUNKLIH 9.4 Ki 5
YIGPWWJHDOXRHC 9.4 Ki 4
VTXIBIOXWRGGBL 9.4 Ki 2
ILFZZMYJRPZIPF 9.4 Ki 5
UZSODGXWZNTIPF 9.3 Ki 3
AZLLXOVNVMQRNP 9.3 Ki 4
XKENJWNGLCKOBP 9.3 IC50 16
UPMDLTAPSSWEPU 9.3 Ki 4
NJUMMJUUDUYSKB 9.3 IC50 16
HLKYSQGBIIIQJN 9.3 Ki 5
SRAWBNFSMIHBEM 9.3 Ki 8
AJTIJRUGVRMRDN 9.3 Ki 5
BPTASZCHRIMWEF 9.3 Ki 6
COIHYICCVMGEJO 9.3 Ki 3
XJRDHPKTMGWJGN 9.3 Ki 6
ZHPXUSDIAXKCGY 9.3 Ki 3
LVJXDIPOLXCUPP 9.3 Ki 3
LDXAQEAQNGTFAB 9.2 Ki 4
VJCYGDVWTVTYGY 9.2 Ki 2
2D structure